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N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-(3-cyclopropyl-5-{3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propyl}-1H-1,2,4-triazol-1-yl)pyridine
1-({1-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4S)-4-(4-ethenylbenzamido)-N-ethyl-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N,N-dimethyl-5-[2-(morpholin-3-yl)acetamido]-1-benzothiophene-2-carboxamide
(2R)-3-(4-chlorophenyl)-2-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamido}propanoic acid
1-ethyl-4-({methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)pyrrolidin-2-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
methyl 1-[2-hydroxy-3-(4-{[(1-methylpiperidin-4-yl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(3-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]acetamide
3-[(3R,4S)-1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-amino-1-{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}pyrrolidine-3-carboxylic acid
1-methyl-N-(4-phenylbutyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-chloro-N,N-dimethyl-3-[({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]imidazo[1,2-a]pyridine-2-carboxamide
1-(1,3-benzothiazol-2-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
5-benzyl-5-{1-[3-(2-oxopyrrolidin-1-yl)benzoyl]piperidin-4-yl}imidazolidine-2,4-dione
1-cyclohexyl-3-methyl-4-(4-methyl-1H-imidazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(2,3-dihydro-1H-inden-2-yl)piperazine
1-[(2-chloro-4-fluorophenyl)methyl]-N-(2,2-dimethyloxan-4-yl)-1H-1,2,3-triazole-4-carboxamide
1-{[1-(4-chlorophenyl)cyclobutyl]methyl}-3-(methoxymethyl)pyrrolidine
4-[2-(pyridin-2-yl)-1H-imidazol-1-yl]thiophene-2-carboxamide
5-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}-N-(propan-2-yl)pyrimidin-2-amine
2-methyl-2-(2-{[1-(methylcarbamoyl)propyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
6-(2-chlorophenyl)-N-ethyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-({3-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}methyl)-4H-chromen-4-one
4-(5-fluoropentyl)-3,4-dihydro-2H-1,4-benzothiazin-3-one
N,N-dimethyl-6-[2-(trifluoromethoxy)phenyl]pyridazin-3-amine
N-[3-(cyclopentyloxy)phenyl]-3-oxo-4-phenylpiperazine-1-carboxamide
1-{2-[3-(3,4-dimethylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}-4-methylpiperazine
1-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3-(pyrrolidin-1-ylmethyl)piperidine
2-{2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-2-oxoethyl}-2-azaspiro[4.4]nonan-3-one
1-[(2-chloro-4-fluorophenyl)methyl]-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
(1R,2R,6S,7S)-4-(3,6-dimethylpyrazin-2-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-ethyl-N-methyl-N-(oxan-2-ylmethyl)pyrimidine-5-carboxamide
(3-{2-[1-(5-fluoro-2-methoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
3-[(3-methoxypyrrolidin-1-yl)sulfonyl]-N-(thiophen-3-ylmethyl)benzamide
1-(pyridin-3-yl)-4-[(3R,5S)-5-(pyrrolidine-1-carbonyl)piperidine-3-carbonyl]piperazine
1-methyl-N-[3-(methylsulfanyl)propyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-(3-methyl-1H-pyrazol-5-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-benzyl-N-methyl-3-[1-(2-phenylpropyl)piperidin-4-yl]propanamide
(cyclohex-3-en-1-ylmethyl)({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
2,8-dimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}quinoline-4-carboxamide
4-amino-N-(3-chloro-4-fluorophenyl)azepane-1-carboxamide
2-[4-(3-chloropyridin-2-yl)-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
3-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
5-ethyl-1'-(quinoxalin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]