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3-methyl-2-[5-(2-methyloxolan-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
2-cyclopentyl-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-[2-(dimethylamino)ethyl]-5-oxo-N-[(4-phenylphenyl)methyl]pyrrolidine-3-carboxamide
2-(morpholin-3-yl)-N-[2-(2-propoxyphenyl)ethyl]acetamide
5-{3-amino-4,6-dimethyl-1H-pyrazolo[3,4-b]pyridin-5-yl}pyridin-3-amine
1-cyclopentyl-N-(2-methoxy-2-methylpropyl)-6-oxopiperidine-3-carboxamide
N-{2-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-oxoethyl}acetamide
8-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-ethyl-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(pyridin-4-ylmethyl)acetamide
N-cyclopentyl-5-[(3-methoxyphenyl)methyl]-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-ethoxy-3-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]pyridine
3-[(dimethylamino)methyl]-1-(2-propylpyridine-4-carbonyl)piperidin-3-ol
2-methyl-2-phenyl-1-[2-(trifluoromethyl)morpholin-4-yl]propan-1-one
(3S,4S)-3-hydroxy-4-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1λ6-thiolane-1,1-dione
(1R,5R)-3-methanesulfonyl-6-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl][1-(pyridin-2-yl)propan-2-yl]amine
5-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
4-[(4-{[1-(4-methylbenzoyl)piperidin-3-yl]methoxy}phenyl)methyl]thiomorpholine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[(3-phenyloxolan-3-yl)methyl]cyclopropanamine
2-{3-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]phenoxy}ethan-1-ol
2-methoxy-N-[(5-{[4-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]acetamide
1-[(2-fluoro-4-methoxyphenyl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
2,3,5-trimethyl-N-[2-(pyridin-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(2,6-dimethylpyridin-3-yl)-3-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]urea
(1S,5R)-6-methanesulfonyl-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-(2-methyl-1H-1,3-benzodiazol-1-yl)-1-(3-phenylpiperidin-1-yl)propan-1-one
6-{4-[4-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}pyridine-3-carbonitrile
3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-5-(3-fluoro-4-methoxyphenyl)-1,2,4-triazine
1-{2-amino-4-[methyl(1H-pyrazol-3-ylmethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-methoxyethan-1-one
3-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-N-(pyridin-3-yl)propanamide
(1R,3R)-N1-{1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}cyclopentane-1,3-diamine
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamide
N-[1-(4-methanesulfonylphenyl)propyl]-4-(pyridin-3-yl)pyrimidin-2-amine
N3-cyclooctyl-4-oxo-N5-[3-(propan-2-yloxy)propyl]-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(2-fluorophenyl)ethan-1-one
(2R,6R)-4-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]benzamide
(2S)-4-methyl-2-phenyl-1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazine
4-{1H-imidazo[4,5-c]pyridin-2-yl}-3-(4-phenylphenyl)-1H-pyrazole
N-[(4,5-dimethylfuran-2-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)-2-(piperidin-1-yl)acetamide
5-{methyl[(3-methyloxetan-3-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-methyl-1-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]-1,4-dihydroquinolin-4-one
3-[(1R,5S)-3,6-diazabicyclo[3.2.2]nonan-6-ylmethyl]-1-methyl-1,2-dihydroquinolin-2-one
4-chloro-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}-1H-pyrrole-2-carboxamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-4-(1H-pyrazol-4-yl)butanamide
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[2-(1H-imidazol-4-yl)ethyl]benzamide
N-[(4-fluorophenyl)methyl]-3-methyl-N-(prop-2-en-1-yl)pyridine-2-carboxamide
(2S,4S)-4-(3-chloro-4-hydroxybenzamido)-N-ethyl-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine-2-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazine