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(3R,4S)-1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-4-(4-methoxyphenyl)pyrrolidin-3-amine
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-oxo-2-phenylacetamide
2-methoxy-N-{[8-(quinolin-7-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
3-amino-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1H-1,2,4-triazole-5-carboxamide
5-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-2,4-dimethylpyrimidine
{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}[(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amine
N-(6-phenoxypyridin-3-yl)-1-(thiophen-3-ylmethyl)piperidine-4-carboxamide
1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
9-(6-phenylpyridazin-3-yl)-1,4,9-triazaspiro[5.5]undecan-5-one
1-(diethylamino)-3-{2-methoxy-5-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)methyl]phenoxy}propan-2-ol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-methyl-5-phenyl-1H-pyrrole-2-carboxamide
1-{1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carbonyl}piperidin-3-ol
8-{[4-(1H-imidazol-1-yl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-oxo-6-[(4-phenylpiperidin-1-yl)methyl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2-dihydropyridine-3-carboxamide
N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)carbamoyl}methyl)piperidine-4-carboxamide
3-{[(cyclopropylmethyl)(2-methoxyethyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(1R,5R)-6-(furan-2-carbonyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
1'-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-chloro-5-[1-(3-methylpyridin-2-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
3-[2-(dimethylamino)ethyl]-5-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]-5-(3-methylbutyl)imidazolidine-2,4-dione
N-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-2-ethylmorpholine-4-carboxamide
ethyl 5-[3-(furan-2-yl)benzoyl]-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-{5-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
6-ethyl-N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
2-{3-[2-(methylsulfanyl)ethyl]-5-[(2-oxo-1,2-dihydropyrimidin-1-yl)methyl]-1H-1,2,4-triazol-1-yl}benzoic acid
1-[2-(2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-1,4-diazepane-6-carboxylic acid
N-[(1-benzylpiperidin-2-yl)methyl]-N-methyloxan-4-amine
5-methyl-N-[2-(pyrazin-2-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
6-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2,4-dimethylpyridine-3-carbonitrile
[1-(4-methoxypyrimidin-2-yl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
N-{1-oxaspiro[4.4]nonan-3-yl}-1-(9H-purin-6-yl)piperidin-4-amine
N-benzyl-2-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}acetamide
3-(1-methylpiperidin-2-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}propanamide
N-benzyl-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}benzene-1-sulfonamide
2-[2-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propanoic acid
2-(pyridin-3-ylmethyl)-8-(1H-1,2,4-triazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]-6-(1-methyl-1H-imidazol-2-yl)pyridazine
2-[(3-chlorophenyl)methyl]-N-[2-(3-hydroxypiperidin-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
5-[4-(2-ethoxyphenyl)piperazin-1-yl]-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-[(7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
1-{3-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-oxopropyl}pyrrolidin-2-one
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
3-methoxy-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
3-(1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-N-(3-methylphenyl)propanamide
N-(2-fluorophenyl)-3-{1-[2-(pyridin-3-yloxy)acetyl]piperidin-3-yl}propanamide
(3S,4R)-1-[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4-(hydroxymethyl)piperidin-3-ol
1-[(2-chlorophenyl)methyl]-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide