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5-[(3S,4S)-3-carboxy-4-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1H-imidazole-4-carboxylic acid
methyl 2-(2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}phenoxy)acetate
N,3,6-trimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1-benzofuran-2-carboxamide
(4aR,8aR)-2-(2-phenoxyethyl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-[(3R,4S)-4-(5-methylfuran-2-yl)-1-(oxan-4-yl)pyrrolidin-3-yl]cyclopropanesulfonamide
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(4-phenyloxan-4-yl)methyl]acetamide
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-(2-phenoxyethyl)piperazine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(prop-2-en-1-yl)piperidine-3-carboxamide
methyl({[3-({1-[4-(4-methylphenyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl})(thiophen-3-ylmethyl)amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-fluoropyridin-2-yl)piperidin-3-ol
7-(1-benzothiophen-3-yl)-4-(pyrimidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-[(3-methoxyphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(pyrimidin-2-yl)ethan-1-one
ethyl 3-[(2-fluorophenyl)methyl]-1-(2-methoxyacetyl)piperidine-3-carboxylate
2-[({2-[3-(azocan-1-yl)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)amino]propane-1,3-diol
(1S,5R)-6-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3-fluorophenyl)methyl]-5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-[4-({[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]carbamoyl}methoxy)phenyl]propanamide
N,N-diethyl-1-[(1s,4s)-4-(3,3-dimethylbutanamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-(2-benzylmorpholin-4-yl)-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
(2R)-2-amino-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-phenylpropan-1-one
3-{5-[(5-methylthiophen-2-yl)sulfonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
4-{[5-(2,5-dimethoxyphenyl)-2-hydroxyphenyl]methyl}piperazine-1-carbaldehyde
1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-methoxy-N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
2,7,8-trimethyl-4-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]quinoline
N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]-1H-indole-2-carboxamide
2-(1-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1-methyl-1H-1,3-benzodiazole
2-(3-{[({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)amino]methyl}-2-methyl-1H-indol-1-yl)acetamide
5-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrazin-2-ol
9-(2,1,3-benzoxadiazol-4-ylmethyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(7-{2-[3-(trifluoromethyl)phenyl]acetyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]oxolane-3-carboxamide
1-methyl-N-[2-(1-methylpiperidin-3-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{2-[7-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-(4-fluorophenyl)acetamide
3-(2-fluorophenyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
N-(2,3-dihydro-1H-inden-4-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
6-{[(cyclopropylmethyl)(propyl)amino]methyl}-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
5-[({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
5-tert-butyl-3-{[4-(1H-imidazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole
6-cyano-N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]pyridine-3-carboxamide
4-phenyl-N-{[1-(1,3-thiazole-5-carbonyl)piperidin-3-yl]methyl}benzamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-(1-methyl-1H-pyrazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-butyl-N-[3-(propan-2-yloxy)propyl]-1,3-benzoxazole-5-carboxamide
2-[2-oxo-2-(3-phenylpiperazin-1-yl)ethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
4-methyl-3-[2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-benzyl-4-[3-(1H-pyrazol-1-yl)propanoyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
4-{[5-(methoxymethyl)thiophen-2-yl]formamido}-N,4-dimethylpentanamide
2-(3-fluorophenoxy)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-1-(propan-2-yl)piperidine-3-carboxamide