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2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
4-(4-benzylpiperazin-1-yl)-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
methyl 6-[2-({[4-(2-oxopyrrolidin-1-yl)phenyl]formamido}methyl)-2,3-dihydro-1-benzofuran-7-yl]pyridine-3-carboxylate
2-(4-methyl-1,4-diazepan-1-yl)-1-(4-phenylazepan-1-yl)ethan-1-one
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-(4-phenoxybenzoyl)piperidine
3-cyclopropyl-1-{4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}urea
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2,4,6-trifluorophenyl)acetamide
N-[3-(3,4-dimethylphenoxy)propyl]-N-methyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N,2-dimethyl-N-{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}propanamide
(3aS,6aS)-2-methanesulfonyl-5-[3-(1H-pyrazol-1-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
2,5-dimethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
7-[2-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]-4-methyl-1,2-dihydroquinolin-2-one
5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-(quinoxalin-6-ylmethyl)-1,2-oxazole-3-carboxamide
2-oxo-1-phenyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidine-3-carboxamide
5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazole
N-methyl-5-(naphthalen-1-yl)-N-(pyridin-3-ylmethyl)-1,2,4-triazin-3-amine
N-benzyl-1-{2-[(2,3-dimethoxyphenyl)formamido]ethyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
3-[2-(4-fluorophenyl)ethyl]-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(2R)-1-{[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl}pyrrolidine-2-carboxamide
6-methyl-N4-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)pyrimidine-2,4-diamine
N,N,4-trimethyl-5-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}pyrimidin-2-amine
N-[2-(phenylsulfanyl)ethyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-3-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}-1,4-dihydropyridin-4-one
N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
{[3-({1-[3-(3-fluorophenyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}(methyl)(thiophen-3-ylmethyl)amine
3-[3-({[3-(pyridin-3-yloxy)propyl]amino}methyl)-1H-indol-1-yl]propanamide
N-{1-[4-(4-phenylpiperazine-1-carbonyl)phenyl]-1H-pyrazol-4-yl}oxolane-3-carboxamide
8-(5-hydroxypyrazine-2-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-{[4-(propan-2-yl)phenyl]methyl}-2-(propane-1-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
3-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1-[4-(1H-1,2,4-triazol-1-yl)phenyl]urea
N-benzyl-2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-(4-chlorophenoxy)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxylic acid
N-{[2-(3-methylphenyl)-6-oxo-1,6-dihydropyrimidin-4-yl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
methyl 3-[(3,4-difluorophenyl)methyl]-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{3-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-3-carboxamide
4-(5-methylpyridin-2-yl)-1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)piperidin-4-ol
7-(3-methoxyphenyl)-2-(3-methylpyridin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(3S,4R)-1-(2,3-difluoro-4-methoxybenzoyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
2-(2,3,4-trimethoxyphenyl)pyridin-4-amine
N4-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-N1,N1-dimethylpiperidine-1,4-dicarboxamide
1-[2-methoxy-5-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol