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4-[5-(dimethyl-1,2-oxazol-4-yl)-3-methyl-1H-1,2,4-triazol-1-yl]-2-methylpyridine
2-methyl-4-oxo-N-(2-phenylphenyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
3-(azepane-1-sulfonyl)-5-(2,4-dimethoxyphenyl)benzoic acid
5-[(2-fluorophenyl)methyl]-5-(1-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
N-(1-{7-[(2-chloro-3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-(1,3-benzothiazol-2-yl)-2-{[2-(hydroxymethyl)piperidin-1-yl]methyl}phenol
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-3-carboxamide
1-(1,2,3,4-tetrahydroisoquinolin-2-yl)-3-[3-(thiomorpholin-4-ylmethyl)phenoxy]propan-2-ol
1-{1-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-2-phenylethan-1-ol
8-[4-(2-fluorophenyl)benzoyl]-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
[1-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl](thiophen-2-yl)methanol
2-[4-(4H-1,2,4-triazol-4-ylmethyl)-1,3-thiazol-2-yl]pyrimidine
N-methyl-N-[2-(4-methylphenoxy)ethyl]-4-oxo-3,4-dihydroquinazoline-2-carboxamide
N-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-6-hydroxy-1,4-oxazepane-4-carboxamide
N-(1-benzothiophen-5-ylmethyl)-9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
3-methyl-4-oxo-N-(1H-pyrazol-3-yl)-3,4-dihydrophthalazine-1-carboxamide
2-(4-{[4-(cyclopentyloxy)phenyl]methyl}piperazin-1-yl)-1-(pyrrolidin-1-yl)ethan-1-one
N-[(2-methoxyphenyl)methyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
3-(2-methylphenyl)-3-phenyl-N-(pyridin-2-ylmethyl)propanamide
2-[methyl(pyridin-2-ylmethyl)amino]-1-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
5-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-4-fluoro-N-(furan-2-ylmethyl)benzamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)furan-3-carboxamide
4-{5-[1-(2-methylfuran-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}morpholine
2-(2-methyl-1,3-thiazol-4-yl)-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}acetamide
(3S,4S)-4-(naphthalen-2-yl)-1-(thiophene-3-carbonyl)piperidin-3-ol
methyl 3-{[2-(2-methylphenyl)acetamido]methyl}-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
(2E)-1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(pyridin-3-yl)prop-2-en-1-one
ethyl 2-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]acetate
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenylethyl)amine
diethyl({4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5-methylfuran-2-yl}methyl)amine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methoxypyrimidin-2-amine
(3-{[1-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
1-[(2-chloro-4-fluorophenyl)methyl]-N-[1-(1H-indol-1-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-tert-butyl-6-(2-methoxy-5-methylbenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-(prop-2-en-1-yl)-9-(2,4,5-trifluorobenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(2-methoxyphenyl)methyl]-6-oxo-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}piperidine-3-carboxamide
methyl[(3-methyl-1H-pyrazol-4-yl)methyl]{[4-(trifluoromethyl)phenyl]methyl}amine
ethyl 2-[2-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,3-thiazole-4-carboxylate
2-[2-(furan-3-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]-1-methyl-1H-1,3-benzodiazole
3-(2-methoxypyridin-3-yl)-1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-(pyridin-4-ylmethyl)urea
1-(furan-3-carbonyl)-4-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1,4-diazepane
2,8-dimethyl-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}quinoline-4-carboxamide
4-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1,4-oxazepane
(3S,4R)-1-[1-(4-methanesulfonylphenyl)cyclobutanecarbonyl]-4-methylpiperidine-3,4-diol
6-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide