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6-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyridine-2-carboxylic acid
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-(1H-indol-1-yl)ethan-1-one
(3S)-1-(2,8-dimethylquinoline-4-carbonyl)-N,N-dimethylpyrrolidin-3-amine
2-methyl-5-(4-{[(6-methylpyridazin-3-yl)amino]methyl}piperidin-1-yl)-2,3-dihydropyridazin-3-one
5-{1-[2-(furan-2-yl)-2-oxoacetyl]pyrrolidin-2-yl}-N-methyl-N-(2-methylpropyl)thiophene-2-carboxamide
4-ethyl-9-(4-oxo-4H-chromen-3-yl)-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinoline-3,7-dione
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-(3-methylphenoxy)ethan-1-one
2-[(2-{1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
3-(2-fluorophenyl)-5-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(2R,6R)-4-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-6-carboxylic acid
methyl 2-{1-[(6,7-dimethyl-2-oxo-2H-chromen-4-yl)methyl]-3-oxopiperazin-2-yl}acetate
N-[(3,4-dimethoxyphenyl)methyl]-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)benzamide
1-(2-methoxyethyl)-8-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(1H-1,3-benzodiazol-2-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)propanamide
2-(4-chlorophenyl)-4-(2-methoxypyrimidine-5-carbonyl)morpholine
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-[(2-phenoxyacetamido)methyl]benzoate
N-[3-(dimethylcarbamoyl)phenyl]-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-{3-[(3-chlorophenyl)methyl]-5-(1H-1,2,3-triazol-5-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-(2,3-difluoro-4-methoxybenzoyl)-3-(2-methylphenyl)piperidine
5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
2-ethoxy-4-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}phenol
8-benzyl-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(1-methyl-1H-pyrazol-5-yl)-N-(pyridin-4-ylmethyl)propanamide
1-(3-{1-[(2-amino-1,3-thiazol-4-yl)methyl]-1H-imidazol-2-yl}-2,4,6-trimethylphenyl)ethan-1-one
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
(3S,9aR)-3-benzyl-2-methyl-8-(quinolin-6-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4S)-4-(propan-2-yl)-3-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,3-oxazolidin-2-one
3-({[1-(2,3-dihydro-1-benzothiophene-2-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
N-[4-(3-methoxyphenyl)phenyl]-1-(oxan-4-yl)pyrrolidine-2-carboxamide
(1R,5S)-6-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
4-(4-methylpiperazin-1-yl)-6-[3-(piperidin-1-ylmethyl)piperidin-1-yl]pyrimidin-2-amine
2-ethyl-9-[(2-ethylpyrimidin-4-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
1-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-oxo-1-phenyl-N-[2-(piperidin-1-yl)ethyl]pyrrolidine-3-carboxamide
1-(2-methoxyphenyl)-N-[2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
(1R,7S)-N-methyl-3-[(3-methylphenyl)methyl]-4-oxo-N-(pyrimidin-4-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[(2-fluorophenyl)methyl]-N-[2-(pyridin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[5-(propan-2-yl)pyrimidin-4-yl]piperidin-3-ol
5-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-methylpyridin-2-amine
N-[(3R,4S)-1-(5-cyanopyridin-2-yl)-4-propylpyrrolidin-3-yl]-3-hydroxypropanamide
(1R,7S)-3-(4-fluoro-2-methylphenyl)-N-methyl-4-oxo-N-(pyrazin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-amino-6-(2H-1,3-benzodioxol-5-yl)-4-(1,2-dimethyl-1H-imidazol-5-yl)pyridine-3-carbonitrile
N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
14-(2-methoxypyrimidin-5-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-[1-(4-fluorophenyl)propyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(4-fluorophenyl)methyl]-3-[1-(2-oxoimidazolidine-4-carbonyl)piperidin-4-yl]propanamide