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N3-(1,3-benzothiazol-2-ylmethyl)-1-benzyl-N5-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(propane-1-sulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2-phenylethyl)-4-[(thian-4-yl)amino]pyrrolidin-2-one
3-[(4-fluorophenyl)methyl]-5-methyl-5-[1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
3-hydroxy-1-[(3-methylphenyl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-2-one
8-[3-(benzylsulfanyl)propanoyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
5-methyl-4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1,3-oxazole
N-[phenyl(thiophen-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
ethyl(methyl)[(5-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]amine
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
4-(4-ethoxy-3-methylphenyl)-N-{[(3R,4R)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}butanamide
1-{[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]amino}cyclopentane-1-carboxamide
(2-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methanol
(3aR,6aS)-2-{[5-(2-fluorophenyl)furan-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole
methyl 3-[(3,5-dimethylphenyl)methyl]-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(4-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidine-1-carbonyl}phenyl)acetamide
1-{1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]azetidin-3-yl}piperidine
1-{1'-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
{[6-(4-ethylpiperazin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}({[4-(trifluoromethyl)phenyl]methyl})amine
4-(azocane-1-carbonyl)-6-fluoro-2-(pyrimidin-5-yl)quinoline
5-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-(2-methylpropyl)-1H-imidazole
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-7-methyl-2-oxo-1H,2H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
N-{2-[(E)-2-(8-hydroxyquinolin-2-yl)ethenyl]phenyl}pyrrolidine-3-carboxamide
3-cyclopentyl-5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
4,5-dimethyl-2-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propyl]-1,3-thiazole
(3R,4S)-1-[5-(methoxymethyl)furan-2-carbonyl]-4-(4-methoxyphenyl)pyrrolidin-3-amine
3-{4-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
ethyl 2-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]amino}acetate
4-methyl-N-[1-(morpholin-4-ylmethyl)cyclopentyl]pyrimidin-2-amine
1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-phenylethan-1-one
3-({2-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
3-[(4-hydroxy-4-phenylpiperidin-1-yl)methyl]-6-methyl-1,2-dihydroquinolin-2-one
1-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]cyclopropan-1-amine
3-(dimethyl-1,2-oxazol-4-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}propanamide
2-[4-(2-phenylethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
6-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-4-(trifluoromethoxy)benzene-1-sulfonamide
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]ethan-1-one
(4aS,8aR)-6-(furan-2-carbonyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(1H-1,3-benzodiazol-2-ylmethoxy)-1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}ethan-1-one
1-(cyclohexylmethyl)-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-2-one
N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
5-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-5-[(2-fluorophenyl)methyl]imidazolidine-2,4-dione
4-[2-(1H-indol-3-yl)acetyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(dimethylamino)-1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}butan-1-one
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
1-{[3-(2,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indazole
N-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}azetidine-1-carboxamide
N,N-bis(2-methylpropyl)-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide