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methyl({[2-(pyrrolidin-1-ylmethyl)phenyl]methyl})(1,3-thiazol-4-ylmethyl)amine
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}urea
methyl 5-{[1-(methylsulfanyl)propan-2-yl]amino}-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
ethyl 4-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-3-yl}piperazine-1-carboxylate
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
N-(furan-2-ylmethyl)-2-{4-[methyl(2-phenylethyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}acetamide
N-({1-[(8-fluoroquinolin-2-yl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]thiophene-2-sulfonamide
5-[1-(1-methylcyclopropanecarbonyl)pyrrolidin-2-yl]-N-[2-(1,3-thiazol-2-yl)ethyl]thiophene-2-carboxamide
{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
2-(2,3-dihydro-1H-isoindol-2-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
5-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)-2-(pyridin-2-yl)pyrimidine
3-(1,3-benzothiazol-5-yl)-1-[(3R)-1-benzylpyrrolidin-3-yl]-1-methylurea
3-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
methyl({[5-(oxolan-2-yl)thiophen-2-yl]methyl}){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
[(3R,4R)-1-(2-ethylbenzoyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-{[2-(dimethylamino)-2-(2-methylphenyl)acetamido]methyl}thiophene-2-carboxylic acid
5-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N-[4-(propan-2-yl)phenyl]-1-(quinoxalin-2-yl)piperidin-3-amine
5-fluoro-N4,N4-dimethyl-N2-[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]pyrimidine-2,4-diamine
3-(1-methyl-1H-pyrazol-4-yl)-1-[2-(pyridin-3-yl)piperidin-1-yl]propan-1-one
methyl 3-(naphthalene-1-carbonyl)-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(2-oxoimidazolidin-1-yl)-N-{[1-(prop-2-en-1-yl)pyrrolidin-3-yl]methyl}benzamide
(1S,5R)-N-[4-ethoxy-3-(trifluoromethyl)phenyl]-10-oxo-3,9-diazabicyclo[3.3.2]decane-3-carboxamide
2-(4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
4-methoxy-2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidine
4-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-1H-pyrazole-3-carboxylic acid
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2,3,4-trimethoxybenzamide
4-chloro-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1,5-dimethyl-1H-pyrazole-3-carboxamide
N-(furan-2-ylmethyl)-2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]acetamide
2-(3-acetyl-1H-pyrazol-1-yl)-N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)acetamide
N-[2-(2-chloro-6-methylphenoxy)ethyl]-1-methylazepane-2-carboxamide
(4aS,8aR)-6-(3-fluoropyridin-2-yl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[1-(7-{[4-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclopropanecarboxamide
3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-[(4-methylphenyl)methyl]piperidine-1-carboxamide
(3S,4S)-1-(1H-imidazol-2-ylmethyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
8-[(2-propoxynaphthalen-1-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
5-{2-benzyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}pyridine-2-carbonitrile
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)cyclohex-3-ene-1-carboxamide
1-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-4-ethylpiperazine-2,3-dione
2-(1-benzyl-3-oxopiperazin-2-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
3-[2-ethoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-6-methylpyridazine
1-[(4-methoxyphenyl)methyl]-4-(2-methyl-1,3-thiazole-5-carbonyl)piperazin-2-one
3-methyl-N-[2-(3-phenylpropoxy)phenyl]-1H-pyrazole-4-carboxamide
2-(1-benzofuran-2-yl)-1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-imidazole
N-(4-cyanophenyl)-4-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]butanamide
1-methyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]azepane-2-carboxamide
4-benzyl-3-ethyl-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
2-(4-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenyl)-5,6-dimethyl-3,4-dihydropyrimidin-4-one