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N-[2-(1H-imidazol-4-yl)ethyl]-6-(methoxymethyl)pyridine-2-carboxamide
8-[(8-methoxyquinolin-2-yl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-[(1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-yl)methyl]pyrrolidin-2-one
methyl 3-chloro-4-{[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)carbamoyl]amino}benzoate
1-(6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-amido)cyclopentane-1-carboxylic acid
1-[3-(2-ethoxyethyl)-4-(morpholin-4-yl)phenyl]ethan-1-one
3-{5-[(4-cyanophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-(2-hydroxyethyl)propanamide
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-phenylpropyl)piperidine
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-({[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
4-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-1-(4-methoxybenzoyl)piperidine
1-{4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-one
(1S,5R)-6-(cyclobutylmethyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(2-hydroxyethyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(2-methoxyphenyl)methyl]piperidine
5-{4-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenyl}-1,3,4-thiadiazol-2-amine
(2S,4R)-4-amino-1-[2-(2,3-dihydro-1H-indol-1-yl)-2-oxoacetyl]-N,N-diethylpyrrolidine-2-carboxamide
4-ethyl-3-{1-[2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S)-N-methyl-4-[(naphthalen-1-ylmethyl)amino]-1-(propan-2-yl)pyrrolidine-2-carboxamide
3-benzyl-4-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperazin-2-one
2-amino-4-(1,5-dimethyl-1H-pyrazol-4-yl)-6-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
N-[3-(2-oxopyrrolidin-1-yl)propyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
2-{[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]methyl}benzoic acid
4-benzyl-3-ethyl-1-[2-(1,3-thiazol-4-yl)ethyl]-1,4-diazepan-5-one
2-cyclopropyl-N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-4-methylpyrimidine-5-carboxamide
2-oxo-8-[3-(1H-pyrazol-1-yl)propyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(2,1,3-benzoxadiazol-5-ylmethyl)pyrazolo[1,5-a]pyridine-7-carboxamide
5-[3-(2-ethylpiperidine-1-carbonyl)-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]quinoline
3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole
3-cyclopropyl-N-[4-(morpholine-4-carbonyl)phenyl]-1H-pyrazole-5-carboxamide
N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(3S,5R)-N3-cyclopropyl-N5-(4-fluorophenyl)-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-{5-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
N-[(3S)-2-oxoazepan-3-yl]-2,2-diphenyl-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}acetamide
1-[cyclohexyl(methyl)amino]-3-(2-{[(2-methoxyethyl)(propan-2-yl)amino]methyl}phenoxy)propan-2-ol
3-[5-(1-benzofuran-5-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-N-cyclopropylpropanamide
3-(2-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-oxoethyl)-3,4-dihydroquinazolin-4-one
3-(1-methylcyclopropyl)-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]propan-1-one
6-(2,3-dihydro-1H-isoindol-2-yl)-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
4-ethenyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
6-methyl-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]imidazo[1,2-a]pyridine-2-carboxamide
2-methoxy-1-{4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(1H-indole-3-carbonyl)piperidin-3-yl]propanamide
5-{2-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-oxoethyl}-2-ethyl-6-methyl-3,4-dihydropyrimidin-4-one
(2S,4S)-4-amino-1-{[2,5-dimethyl-1-(pyridin-3-yl)-1H-pyrrol-3-yl]methyl}-N-methylpyrrolidine-2-carboxamide
1-(cyclobutylmethyl)-3-hydroxy-3-({[(6-methylquinolin-5-yl)methyl]amino}methyl)piperidin-2-one
N-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}methyl)pyridine-2-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-ethyl-4-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide