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4-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-6-(propan-2-yl)pyrimidine
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-ethyl-5-methyl-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)thiophene-3-carboxamide
2-(1H-1,2,3-benzotriazol-1-yl)-N-(1-ethyl-1H-indazol-3-yl)acetamide
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]benzamide
N-[(2S)-1-hydroxypropan-2-yl]-5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carboxamide
2-{2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
(2R,6R)-10-methoxy-4-(6-methyl-2-propylpyrimidin-4-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-4-(hydroxymethyl)azepan-4-ol
1-{1'-[2-(2-fluorophenyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
(1R,5S)-6-methyl-3-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3-cyclopentylpropyl)-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
(1S,5R)-6-benzyl-3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-hydroxy-2-(1-methyl-1H-imidazol-2-yl)ethyl]-1,2,3,4-tetrahydronaphthalene-2-carboxamide
1-(2-ethoxyethyl)-4-(2-methyl-1-benzofuran-5-carbonyl)piperazine
N-cyclobutyl-3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
4-[5-(pyrimidin-5-yl)furan-2-carbonyl]morpholine
2-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-4-yl}-1-methyl-1H-1,3-benzodiazole
N-cyclopropyl-N-{[4-(thiophen-3-ylmethoxy)phenyl]methyl}quinoline-2-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
N-benzyl-2-{1-oxo-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-2-yl}-N-(1,3-thiazol-2-ylmethyl)acetamide
7-{[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-4-methyl-2H-chromen-2-one
2-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]urea
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[(1-propyl-1H-imidazol-2-yl)methyl]-decahydro-2,7-naphthyridine-2-sulfonamide
2-{1-cyclohexyl-4-[(6-ethoxyquinolin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(1S,5R)-6-[2-(3-methoxyphenoxy)ethyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
4-{2-ethyl-3H-imidazo[4,5-b]pyridin-6-yl}-1-methyl-1H-pyrrolo[2,3-b]pyridine
1-{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-2,2-bis(prop-2-en-1-yl)piperidine
1,4-dimethyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidine-4-carboxamide
2-[(cyclopropylmethyl)sulfanyl]-1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]ethan-1-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
1-[(4-methyl-1H-imidazol-5-yl)methyl]-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
1-[(1-{6-[benzyl(methyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
4-(3-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carbonyl)morpholine
N-cyclopropyl-3-{1-[(3-ethoxyphenyl)methyl]piperidin-3-yl}propanamide
2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanamide
5-{1-[(2,4-dimethylphenyl)methyl]piperidin-4-yl}-5-[(3-methoxyphenyl)methyl]-3-methylimidazolidine-2,4-dione
methyl 4-{[(2-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
2-{4-[(6-chloro-4-hydroxyquinolin-2-yl)methyl]-1,4-diazepan-1-yl}-N,N-dimethylacetamide
2-[(3-fluorophenyl)methyl]-4-(4-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}piperidin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
(3S,4S)-1-[(5-acetylthiophen-3-yl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
2-[(1S,4S)-5-(3-chlorophenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]-N-(1,5-dimethyl-1H-pyrazol-4-yl)acetamide
(1H-imidazol-2-ylmethyl)(methyl)[(3-{[1-(naphthalene-1-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
2-(4-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrazine
4-[2-(dimethylamino)-2-(2-fluorophenyl)acetyl]-1-(3-methoxyphenyl)piperazin-2-one
(1S,5R)-3-[(3,5-difluorophenyl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
6-methoxy-2-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-methyl-2-(phenylsulfanyl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-{[1-(quinoxaline-6-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid