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{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
1-(4-fluorophenyl)-4-[2-(morpholin-4-ylmethyl)piperidin-1-yl]butan-1-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-4-(piperidin-1-ylmethyl)benzamide
2-(cyclopropylmethyl)-8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl 5-{[(3-ethoxy-4-methoxyphenyl)methyl]amino}-1-(2-methoxyethyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
7-chloro-4-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
2-(1H-imidazol-2-yl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]benzamide
(2R)-2-amino-N,4-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pentanamide
{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}(thiophen-3-ylmethyl)amine
(5-{[2-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-2-ethoxyphenyl)methanol
2-[(adamantan-1-ylmethyl)({[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
N-(5-chloro-2-methoxyphenyl)-3-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}propanamide
1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3-(3-methylphenoxymethyl)piperidine
dimethyl({2-[1-(2-methyl-4-phenylpyrimidine-5-carbonyl)piperidin-2-yl]ethyl})amine
2-({[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-6-ethoxyphenol
2-methyl-4-{3-[4-(oxolan-2-ylmethyl)piperazine-1-carbonyl]phenyl}butan-2-ol
2-(pyridin-4-yl)-5-[4-(pyridin-4-yl)piperazine-1-carbonyl]pyrimidine
9-(1-methyl-1H-pyrrole-2-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{3-cyclopentyl-5-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}benzoic acid
(1S,5R)-6-[(4-chloro-3-fluorophenyl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-methyl-7-(7-methyl-4-oxo-4H-chromene-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)(4,4,4-trifluorobutyl)amine
2-{2-[1-(3-methoxypyrazin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(3,5-dimethylphenyl)-4-[(4-methyl-1H-imidazol-5-yl)methyl]piperazin-2-one
1,3-dimethyl-4-{8-methyl-2-[2-(methylamino)pyrimidin-5-yl]quinoline-4-carbonyl}piperazin-2-one
1-(1-methyl-1H-pyrrol-2-yl)-2-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethane-1,2-dione
3-(3-fluoro-4-methoxyphenyl)-4-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-(2-methylphenyl)-1H-pyrazole
methyl 2-[(2-phenylethyl)sulfamoyl]-6-(1,2,3-thiadiazole-4-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-ethyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-yl}-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-({3-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-indole
1-{[3,4-dimethoxy-5-(prop-2-en-1-yl)phenyl]methyl}-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
2-(4-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}morpholin-3-yl)-N-methylacetamide
(1S,5R)-3-(3-phenylpropyl)-6-(1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
2-[3-(3-fluorophenoxymethyl)-5-(2-methyl-4,5,6,7-tetrahydro-2H-indazol-3-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-methyl-2-(propan-2-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1,3-benzoxazole-5-carboxamide
5-butyl-1-(2-methoxyphenyl)-4-[(2-methyl-1,3-oxazol-4-yl)methyl]piperazin-2-one
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-(4-fluorophenyl)acetamide
5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]-1-(3-phenylpropyl)piperidin-2-one
2-[2-(2,5-dioxoimidazolidin-1-yl)acetamido]-2-[2-(trifluoromethyl)phenyl]acetic acid
methyl (2S,4R)-4-(quinoline-2-amido)-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]pyrrolidine-2-carboxylate
ethyl 4-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]piperidine-1-carboxylate
1-(methoxymethyl)-N-[(3R,4S)-4-(propan-2-yl)-1-(pyridin-4-yl)pyrrolidin-3-yl]cyclobutane-1-carboxamide
6-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-9H-purin-2-amine
5-methoxy-1-methyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1H-indole-2-carboxamide
3-({[(2-chlorophenyl)methyl]amino}methyl)-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
5-(2-methoxyphenoxymethyl)-3-(2-phenylazetidine-1-carbonyl)-1H-pyrazole