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1-(2-{[(1-methyl-3-phenyl-1H-pyrazol-5-yl)carbamoyl]amino}ethyl)piperidine-3-carboxamide
4-methyl-2-(pyridin-3-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrimidine-5-carboxamide
(3S,5S,9S)-5-{[(3-chlorophenyl)methyl]amino}-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,4,5-trimethoxybenzamide
3-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
N-[(6-hydroxypyrimidin-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-acetyl-N-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-1,4-diazepane-1-carboxamide
3-(2-ethyl-1H-1,3-benzodiazol-6-yl)-1-methyl-1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]urea
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
2-(2,5-dioxoimidazolidin-1-yl)-N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]acetamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[3-(methylsulfanyl)propyl]propanamide
3-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
N,N-dimethyl-6-(quinolin-3-yl)pyridazin-3-amine
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2H-1,3-benzodioxole-5-carboxamide
methyl 3-(cyclopropylmethyl)-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-({[(2-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
2-[4-(propan-2-yl)phenyl]-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
(3aR,6aR)-2-(3-methylpyrazin-2-yl)-5-(propan-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[6-(2,4,6-trimethylphenyl)pyridin-3-yl]ethan-1-one
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pent-4-en-1-one
1-{4-[2-(4-methylphenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
N,N-dimethyl-6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyrazin-2-amine
methyl (2S,4S,5R)-4-(azepane-1-carbonyl)-1,2-dimethyl-5-phenylpyrrolidine-2-carboxylate
1-cyclohexyl-6-(pyridin-3-ylmethoxy)-4-[4-(thiophen-2-yl)butanoyl]-1,4-diazepan-2-one
dimethyl(2-{2-[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
N-{[4-(3-methoxyphenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
6-(4-{[(1-benzyl-1H-pyrazol-4-yl)methyl]amino}piperidin-1-yl)pyridine-3-carbonitrile
4-[(4-fluorophenyl)methyl]-1-(5-hydroxypyridine-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
4-[4-(2,2-dimethyloxane-4-carbonyl)piperazin-1-yl]benzonitrile
6-methyl-2-(piperidin-1-yl)-N-[1-(pyridin-4-yl)propan-2-yl]pyrimidin-4-amine
N-(1-phenyl-1H-pyrazol-5-yl)-2-(1H-1,2,4-triazol-1-yl)acetamide
3-(6-hydroxy-1,4-oxazepane-4-carbonyl)-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
1-[(3-methoxyphenyl)methyl]-4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperazin-2-one
2-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(1R,7S)-3-tert-butyl-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
2-ethyl-5-({4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyrimidine
8-methyl-2-(1,3-thiazol-5-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
7-(propan-2-yl)-2-(5,6,7,8-tetrahydroquinoline-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-cyclohexyl-N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-pyrazole-4-carboxamide
4-(5-methyl-1,2,4-oxadiazol-3-yl)-1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidine
3-methyl-N-({3-methyl-7-[2-(4-methylphenoxy)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-carboxamide
(3aS,6aR)-5-[(2-fluoro-5-methylphenyl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
[1-({1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
1-(2-fluoro-6-methoxybenzoyl)-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]azocane
methyl 4-{[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]methyl}thiophene-2-carboxylate
methyl 2-{[5-(4-fluorophenyl)-4-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]pyrimidin-2-yl]sulfanyl}acetate