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9-(4-fluorobenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-[(3,5-dimethoxyphenyl)methoxy]-4-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-1-(propan-2-yl)-1,4-diazepan-2-one
2-(4-fluorophenyl)-1-[(1R,5S,8R)-8-hydroxy-3-azabicyclo[3.2.1]octan-3-yl]ethan-1-one
N-{[4-(2-methylpropyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-3-(2-oxoimidazolidin-1-yl)benzamide
(4aS,7aR)-1-(3-hydroxypropanoyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,3,5-trimethyl-N-[(3R,4R)-4-(4-methylpiperazin-1-yl)oxolan-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine
(2-oxo-2-{3-oxo-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}ethyl)urea
8-[4-(trifluoromethyl)benzenesulfonyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[4-(4-{[(2,3-difluorophenyl)formamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-(methoxymethyl)thiophene-2-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)furan-2-carboxamide
N-benzyl-N-ethyl-3-(4-methyl-1,4-diazepan-1-yl)propanamide
4-[1-(5-methyl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]-1-(2-phenylethyl)piperidine
1-cyclopropyl-5-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
2-(5-{1-[(1R,3S,4S)-3-hydroxy-4,7,7-trimethylbicyclo[2.2.1]heptane-1-carbonyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(propan-2-yloxy)propanamide
3-(3-methyl-1H-1,2,4-triazol-1-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
4-(6-methoxyhexanoyl)-1-phenylpiperazin-2-one
2-({[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl](methyl)amino}methyl)-3,4-dihydroquinazolin-4-one
2-[1-(1H-pyrazole-4-carbonyl)piperidine-3-carbonyl]pyridine
3-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3R,4R)-1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(hydroxymethyl)piperidin-3-ol
4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-2-(2,2-diphenylethyl)morpholine
ethyl 1-(1,3-benzothiazol-2-yl)-5-[(3-hydroxypiperidin-1-yl)methyl]-1H-pyrazole-4-carboxylate
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-5-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
N5-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-N6-(2-methoxyethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-(1-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-fluorobenzamide
3-methyl-6-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridazine
1-(3,5-dimethylphenyl)-4-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperazin-2-one
3-[2-(2,2-diphenylethyl)morpholin-4-yl]-N,N-dimethylpropanamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-[(1S,5R)-3-(3-hydroxy-2-methylbenzoyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N,2,8-trimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]quinoline-4-carboxamide
N-(2-hydroxyethyl)-1-methyl-2-oxo-6-(propan-2-yl)-N-(1,3-thiazol-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(pyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-(4-{1-[2-(2-hydroxyethoxy)ethyl]-1H-imidazol-2-yl}phenyl)acetamide
1-(2-phenylpropyl)-3-[4-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
2-(3,4-dichlorophenyl)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]morpholine
N-[2-(4-chlorophenyl)ethyl]-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-(2,3-dihydro-1H-inden-1-yl)-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(2S)-oxolan-2-ylmethyl]-1,2-oxazole-3-carboxamide
5-{[3-hydroxy-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonitrile
1-(cyclopropylmethyl)-N-(pyridin-2-ylmethyl)-5-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-cyclopentyl-4-{[(4,6-dimethylpyrimidin-2-yl)(methyl)amino]methyl}pyrrolidin-2-one
4-[3-(ethanesulfonyl)phenyl]-1-methyl-1H-pyrazole
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-(oxolan-2-ylmethyl)-N-propylpropanamide
5-methoxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-4-oxo-4H-pyran-2-carboxamide
1-[5-(3,5-dimethyl-1H-pyrazol-4-yl)-1H-1,3-benzodiazol-2-yl]ethan-1-ol
5-[1-(2,2-dimethylpropyl)pyrrolidin-2-yl]-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]thiophene-2-carboxamide
2-cyclobutyl-1-methyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-7-(oxolane-2-amido)-1H-1,3-benzodiazole-5-carboxamide
1-({5-[3-(3-fluorophenyl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)-4-methylpiperazine