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2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
3-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
1-benzyl-4-[1-(2-fluorophenyl)cyclopropanecarbonyl]-1,4-diazepan-6-ol
methyl (2S,4R)-1-methyl-4-[3-(trimethyl-1H-pyrazol-1-yl)propanamido]pyrrolidine-2-carboxylate
5-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,3-dimethyl-1H-pyrazole
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(5-propylfuran-2-yl)methyl]piperidine
(2-methoxy-5-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}phenyl)methanol
N-(furan-3-ylmethyl)-N-methyl-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}acetamide
7-[3-(2,4-difluorophenyl)propanoyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(1-benzyl-1H-imidazol-5-yl)methyl]-4-(hydroxymethyl)azepan-4-ol
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-amine
(2S,3R)-3-(3-benzyl-1H-1,2,4-triazol-5-yl)-N-(prop-2-en-1-yl)bicyclo[2.2.1]heptane-2-carboxamide
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
9-(5-methyl-1,3,4-oxadiazol-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-(2-phenylethyl)-1,3-oxazole-4-carboxamide
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-2,5-dimethylpyrimidin-4-amine
7-methyl-3-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
4-(benzenesulfonyl)-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-ethyl-8-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
5-[(3,4-difluorophenyl)methyl]-3-(1-methyl-1H-imidazol-4-yl)-1,2,4-oxadiazole
1-(azepan-1-yl)-3-[2-methoxy-4-({[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]pyridin-3-ol
N'-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-N-(5-methyl-1,2-oxazol-3-yl)ethanediamide
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
1-{2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propyl}-1H-pyrazole
2-(2,5-dioxoimidazolidin-1-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
[1-(1,3-benzothiazol-2-ylmethyl)-4-(oxan-2-ylmethyl)piperidin-4-yl]methanol
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]furan-3-carboxamide
2-cyclopropyl-4-hydroxy-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carboxamide
ethyl 1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-(2-methoxyethyl)piperidine-3-carboxylate
7-(3-chlorophenyl)-4-[(2-fluoro-4-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
N-{[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
9-(2-methoxyethyl)-1-methyl-4-[(5-methylthiophen-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
7-ethyl-N-[(2-fluorophenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
4-(8-methoxyquinolin-5-yl)-N-methylbenzamide
4-[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]-6-(propan-2-yloxy)pyrimidin-2-amine
4-{[(4aS,7aR)-4-cyclobutanecarbonyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzonitrile
2-(morpholin-3-yl)-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethan-1-one
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
methyl 3-(2-methylpropanamido)-6-{spiro[indene-1,4'-piperidine]-1'-ylmethyl}thieno[2,3-b]pyridine-2-carboxylate
N-ethyl-4-formyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}benzamide
{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)(thiophen-2-ylmethyl)amine
3-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
8-[(3-carboxy-4-methoxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[4-(4-chlorophenoxy)piperidine-4-carbonyl]imidazolidin-4-one
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-3-(2-methylphenyl)-3-phenylpropanamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-benzyl-N-(2-hydroxyethyl)propanamide