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methyl (2S,4S,5R)-4-[cyclohexyl(methyl)carbamoyl]-1,2-dimethyl-5-phenylpyrrolidine-2-carboxylate
N-methyl-N-[1-(pyridin-3-yl)propyl]-2-(2,3,4-trifluorophenyl)acetamide
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-oxo-1,3-oxazolidine-4-carboxamide
N-[(5-chlorothiophen-2-yl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
1-butyl-5-(5-chloro-2,3-dimethoxyphenyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
1-methyl-4-[2-(2-methylphenyl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
5-{1-[4-(4-methoxyphenyl)-4-oxobutanoyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
3-{1-[(1-pentylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-1-ol
9-(2-acetylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 3-({4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxyphenyl}formamido)propanoate
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(1-{[1-(propane-1-sulfonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
3-(2-chlorophenyl)-N-(1H-1,2,4-triazol-3-yl)pyrrolidine-1-carboxamide
3-(2,5-dimethoxyphenyl)-1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidine
1-{2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetyl}piperidine-3-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
(2S)-2-(dimethylamino)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-3-phenylpropan-1-one
N-(4-fluoro-2-methylphenyl)-2-{[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}propanamide
N-methyl-N-{1-[1-(pyridin-4-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}thiophene-2-carboxamide
2-[(3-fluorophenyl)methyl]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]morpholine
(2R)-2-methyl-1-{3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]benzoyl}piperazine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-4-(piperidin-1-ylmethyl)benzamide
3-(4-{1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}pyridin-2-yl)phenol
(2R)-2-amino-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
3-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-1-(3,4-dihydro-2H-1-benzopyran-3-yl)urea
N-(2-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methylurea
(1S,5R)-3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
{1-[({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]cyclopropyl}methanol
2-(1,4-dithiepan-6-yl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N,1-dimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(3,5-dimethylbenzoyl)-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(3-{[2-(propan-2-yl)-2,5-dihydro-1H-pyrrol-1-yl]sulfonyl}benzoyl)piperazine
N-methyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
(3S,4S)-N-benzyl-3-hydroxy-4-(propan-2-yloxy)pyrrolidine-1-sulfonamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)-2-(thiophen-3-yl)acetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[3-(1H-pyrazol-1-yl)propyl]amine
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-ol
(4R,6S)-4-methyl-6-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1,3-diazinane-2-thione
4-{4-[(2-methoxypyridin-3-yl)methyl]piperazin-1-yl}-6-methylpyrimidin-2-amine
N-[3-(1,3-thiazol-4-yl)phenyl]-1-[(trimethylpyrazin-2-yl)methyl]piperidine-4-carboxamide
3-{2-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-(4-methylphenyl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}methanesulfonamide
4-chloro-N-[1-(4-fluorophenyl)-2-hydroxyethyl]-1-methyl-1H-pyrazole-3-carboxamide
3-(3-hydroxy-1,2-oxazol-5-yl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
3-(2-hydroxyphenyl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
N-(2,2-dimethyloxan-4-yl)-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide