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3-methyl-7-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3,4-dihydro-2H-1-benzopyran-6-carboxamide
2-[4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)phenoxy]acetic acid
8-(2H-1,3-benzodioxol-5-ylmethyl)-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}morpholin-3-yl)methanol
1-(carbamoylmethyl)-N-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}piperidine-4-carboxamide
1'-(2-ethoxypyridine-3-carbonyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[2-(morpholine-4-carbonyl)piperazin-1-yl]butan-1-one
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-3-ol
1-[(4aR,8aR)-4a-hydroxy-7-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
(2S,4R)-N-ethyl-1-(3-methylbut-2-en-1-yl)-4-{5-[(methylsulfanyl)methyl]furan-2-amido}pyrrolidine-2-carboxamide
2-{4-[(2,6-dimethoxyphenyl)methyl]-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(2-methoxyphenoxy)-N-({1-[2-(phenylsulfanyl)acetyl]piperidin-3-yl}methyl)acetamide
methyl 5-[(2-aminopyrimidin-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-{1-[3-(1H-indol-3-yl)propanoyl]piperidin-3-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
5-(5-chloro-2-fluorobenzoyl)-1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
2-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}-6-methylpyridine
1-methyl-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopropane-1-carboxamide
1-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl 2-(azepane-1-sulfonyl)-6-[(4-ethoxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-methyl-5-(4-{[3-(trifluoromethyl)phenyl]methyl}piperazine-1-carbonyl)pyrimidine
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
N-(1-methyl-1H-indazol-3-yl)-2-[3-(pyridin-4-yl)-1H-indazol-1-yl]acetamide
4-(2-methoxyphenyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanamido]-N-(2-ethylphenyl)benzamide
2-[(3-{[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]carbamoyl}phenyl)amino]acetic acid
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-1-(4-methylphenyl)cyclopropane-1-carboxamide
4-[5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carbonyl]thiomorpholine
2-(5-oxo-1-phenyl-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)-N-[2-(pyrazin-2-yl)ethyl]acetamide
9-methoxy-3-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-N-(3-methylbutyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]-2-(trifluoromethyl)morpholine
5-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2-dihydropyridin-2-one
1-(3-chloro-4-fluorophenyl)-4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazine
3-(methylsulfanyl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]propanamide
4-(5-methylpyridin-2-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-4-ol
1-methyl-4-{1-[1-(1,2-oxazole-3-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
N-[2-(ethanesulfonyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-methyl-N-[(2R)-3-methylbutan-2-yl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-{1-[(6-methylquinolin-5-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
2-(dimethylamino)-N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
4-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)-1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
5-phenyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
4-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2,6-dimethylpyridine
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]but-3-enamide
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(ethylamino)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]pyrimidine-5-carboxamide