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N,N-diethyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carboxamide
diethyl({3-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
(2S,4R)-N,N-diethyl-4-(6-methyl-4-oxo-4H-pyran-2-amido)-1-(propan-2-yl)pyrrolidine-2-carboxamide
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(pyrrolidine-1-carbonyl)piperidine
2-(4-ethylpiperazin-1-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}acetamide
4-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2,6-dimethoxypyrimidine
4-[1-(4,7-dimethylquinazolin-2-yl)piperidine-3-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(3-methoxypropyl)-8-(9H-purin-6-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)benzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-[1-methyl-5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
6-(benzyloxy)-4-(but-2-ynoyl)-1-cyclohexyl-1,4-diazepan-2-one
1-(adamantan-2-ylmethyl)-5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
N-[2-(dimethylamino)ethyl]-3-methyl-N-(thiophen-3-ylmethyl)benzamide
3-(4-methoxyphenyl)-1-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}propan-1-one
2-(3-{9-oxa-2-azaspiro[5.5]undecan-2-ylmethyl}phenoxy)ethan-1-ol
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(3-methylthiophen-2-yl)methyl]furan-2-carboxamide
2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetic acid
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-N-(pyridin-3-ylmethyl)acetamide
ethyl 2-(4-{[2-(3-methoxyphenyl)azetidine-1-carbonyl]amino}phenyl)acetate
4-{[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl]oxy}-3-chloro-N-(2-methoxyethyl)benzamide
N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(pyridin-3-yl)-N-{[7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}propanamide
1-({3-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-1,3-benzodiazole
N-ethyl-N-(2-methylprop-2-en-1-yl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N,1-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
9-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
2-[2-(butan-2-yl)phenoxy]-N-(pyridin-2-ylmethyl)acetamide
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-3-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)urea
3-({2-[1-(propane-2-sulfonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
3-[(2,4,6-trimethylphenyl)methyl]-3,9-diazaspiro[5.6]dodecan-10-one
N-[2-methyl-3-(pyrrolidin-1-yl)phenyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
2-[3-(dimethylamino)propyl]-3-oxo-N-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
5-{3-[4-(furan-2-carbonyl)piperazin-1-yl]-3-oxopropyl}-5-[(4-methylphenyl)methyl]pyrrolidin-2-one
[(3R,4R)-1-(4-chloro-3-fluorobenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-(1-benzofuran-2-ylmethyl)-3-(2,4-dimethoxybenzoyl)piperidine
3-(2,6-dimethoxypyridin-3-yl)-1-[1-(pyrazin-2-yl)propan-2-yl]urea
2-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)-4-phenylphenol
3-[ethyl({[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl})amino]-1λ6-thiolane-1,1-dione
(1S,5R)-3-(6-cyclopropylpyrimidin-4-yl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[1-(1-phenylethyl)-1H-pyrazol-5-yl]-1-[(3-propyl-1,2-oxazol-5-yl)methyl]urea
(1R,5S,6R,7S)-6-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-3-methyl-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-(1-{7-[(3-ethoxy-2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
5-(2-butoxy-4-fluorophenyl)-1-methyl-1H-imidazole
2-[4-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)morpholin-3-yl]-N-phenylacetamide
2-(1H-1,3-benzodiazol-2-ylmethoxy)-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
4-chloro-N-(2-methoxybutyl)-2-propanamidobenzamide
4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrimidin-2-amine