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1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole
2-methyl-5-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-1,3-benzodiazole
N-[2-(dimethylamino)ethyl]-3-acetamido-N-[(2-methylphenyl)methyl]propanamide
3-(2-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](ethyl)amino}-1-hydroxyethyl)phenol
3-(4-chloro-2-methylbenzoyl)-1-(1H-pyrazol-3-ylmethyl)piperidine
3-{4-[3-(methoxymethyl)pyrrolidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}-1H-pyrazole
2-(3-fluorophenoxymethyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]-1,3-oxazole-4-carboxamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
3-fluoro-N-[(2R,3R)-2-methoxy-1'-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
2-amino-1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-methylpropan-1-one
1-(1-benzofuran-2-ylmethyl)-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
3-{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}pyridine
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylpyridin-2-amine
4-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,3-thiadiazole
6-{3-[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(4-methoxypyrimidin-2-yl)piperidine-4-carboxylic acid
2-(3-hydroxyphenyl)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
6-(2,3-dihydro-1-benzofuran-2-carbonyl)-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-2-(2,5-dioxoimidazolidin-4-yl)-N-(2-hydroxyethyl)acetamide
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-4-(1H-1,2,4-triazol-3-yl)benzamide
1-(3-chloro-2-methylphenyl)-3-[1-(methoxymethyl)cyclopentyl]urea
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
N,N-diethyl-1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
4-(3-methylphenoxy)-1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{imidazo[1,2-a]pyrazin-3-ylmethyl}furan-2-carboxamide
9-cyclooctyl-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(3-methoxyphenyl)-4-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperazin-2-one
N5-methyl-N5-[(2-methyl-1,3-thiazol-4-yl)methyl]-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-2-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazole
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-3-(1-methylpiperidin-3-yl)propanamide
1-(4-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}phenyl)-3-methylurea
1-{[5-(4-chlorophenyl)furan-2-yl]methyl}-3-[(dimethylamino)methyl]piperidin-3-ol
2-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
ethyl 5-{[(cyclohexylmethyl)amino]methyl}-1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-1H-pyrazole-4-carboxylate
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-(oxan-4-yl)acetamide
(3S,9aR)-8-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-2-methyl-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
9-(3,5-dimethyl-1H-indole-2-carbonyl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
ethyl 5-{[(1-benzylpiperidin-4-yl)amino]methyl}-1-(4-methylphenyl)-1H-pyrazole-4-carboxylate
4-(4-methoxybenzenesulfonyl)-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
{[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl})amine
2-{1-[(3-methoxyphenyl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
(1S,5R)-3-cyclobutanecarbonyl-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-methyl-2-{2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}pyrrolidine
N-[1-(furan-2-yl)ethyl]-9-methoxy-3-(2-methoxybenzoyl)-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(pyrimidin-2-yl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]piperidin-4-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
N-(2-{5-methyl-4-[(5-phenylpentanamido)methyl]-1,3-oxazol-2-yl}phenyl)pyridine-3-carboxamide
N-[(2R,3R)-1'-(2,3-dihydro-1H-inden-2-yl)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide