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1-[1-(cyclohexylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-ol
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(2S)-2-[(6-methoxypyrimidin-4-yl)amino]-3-phenylpropanamide
(3R,5S)-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
4,6-dimethyl-2-(thiophen-3-yl)pyridine-3-carboxamide
8-(2,2-dimethylpropyl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S)-2-amino-1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-3-(1H-imidazol-4-yl)propan-1-one
(4aR,8aR)-7-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
2-(2-{[4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}phenoxy)acetic acid
N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-4-ylsulfanyl)acetamide
2-[4-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)phenyl]ethan-1-ol
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-[2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1R,5R)-6-(1H-imidazol-2-ylmethyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
[2-(diethylamino)ethyl]({[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl})methylamine
5-acetyl-N-{1-[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]-1H-pyrazol-4-yl}thiophene-2-carboxamide
ethyl 1-[(2H-1,3-benzodioxol-5-yl)carbamoyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(furan-2-yl)propanamide
1-{3-[(1R,3S,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
1-(9H-purin-6-yl)-4-(1H-pyrrole-3-carbonyl)-1,4-diazepan-6-ol
{[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl}(2-phenylpropyl)amine
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
2-{1-[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
4-({4-[3-(diethylamino)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)piperazine-1-carboxamide
2-benzyl-5-(4-fluoro-2-methylbenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine
methyl 3-{[5-(methoxymethyl)furan-2-yl]methyl}-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-(3,4-dimethylphenoxymethyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
5-oxo-1-(pyridin-4-ylmethyl)-N-[2-(2,4,6-trimethylphenyl)ethyl]pyrrolidine-3-carboxamide
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-(pyridin-2-ylmethyl)propanamide
5-(methoxymethyl)-N-[(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]furan-2-carboxamide
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
1-[3-({3-[3-(methoxymethyl)piperidine-1-carbonyl]-1H-pyrazol-5-yl}methoxy)phenyl]ethan-1-one
1-(4-fluorophenyl)-4-{[4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}piperazine
(3aR,6aS)-5-methyl-4,6-dioxo-N-[2-(piperidin-1-ylmethyl)phenyl]-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
1-amino-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}cyclobutane-1-carboxamide
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-2-[2-(2-phenylethyl)pyrrolidin-1-yl]pyrimidine
(2S)-2-[4-(4-chlorophenyl)butanamido]-3-(4-hydroxyphenyl)propanoic acid
methyl 3-{[9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]sulfonyl}thiophene-2-carboxylate
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-4-methyl-1H-imidazole-5-carboxamide
3-(naphthalene-1-carbonyl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
1-[(4-phenyloxan-4-yl)methyl]-5-[2-(propylamino)ethyl]pyrrolidin-2-one
4-(1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)thiomorpholine
3-{[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl](methyl)amino}-N-(pyridin-3-yl)propanamide
1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]propanamide
N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-5-phenyl-1,2-oxazole-3-carboxamide
N2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N4-methyl-5H,6H,7H-cyclopenta[d]pyrimidine-2,4-diamine
4-(pyridin-3-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]pyrimidin-2-amine
(1R,5R)-6-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide