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N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]thiophene-2-carboxamide
1-[3-(1,3-thiazol-4-yl)phenyl]-N-[2-(thiophen-2-yl)ethyl]piperidin-4-amine
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)(quinolin-4-ylmethyl)amine
N-(pyridin-3-ylmethyl)-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
{2-[4-(1H-pyrazol-5-yl)phenyl]pyridin-4-yl}methanol
1-[2-(2,3-dimethylphenoxy)ethyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
4-(4-chlorophenyl)-1-[3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidin-4-ol
2-(4,6-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)acetamide
4-phenoxy-1-[3-(thiophen-2-yl)propanoyl]piperidine-4-carboxylic acid
3-[1-(methoxymethyl)cyclopropyl]-3-methyl-1-(2-methylnaphthalen-1-yl)urea
4-chloro-N,N-diethyl-3-[2-(1H-1,2,4-triazol-1-yl)propanamido]benzamide
2-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1-(2-methoxyethyl)-1H-imidazole
(3aS,6aS)-2-cyclohexyl-5-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(furan-2-ylmethyl)pyrrolidin-3-yl]-2-(methylamino)pyridine-4-carboxamide
3-[5-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]-1-methyl-1-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]urea
2-(1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-3-yl)ethan-1-amine
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl){[5-(oxan-2-yl)furan-2-yl]methyl}amine
5-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-methyl-1H-indazole
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
N-{2-[(2S)-5-oxopyrrolidine-2-carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-1-phenylcyclopropane-1-carboxamide
1-methyl-4-{2-[2-(trifluoromethyl)phenyl]pyridine-4-carbonyl}piperazine
N-({3-methyl-7-[2-(4-methylphenoxy)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-phenylmethanesulfonamide
N-{[7-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine-2-carboxamide
6-oxo-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
5-(furan-2-ylmethyl)-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(4aS,8aR)-1-(2-aminoethyl)-6-(2H-1,3-benzodioxole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1,7-dimethyl-1H-indole-2-carboxamide
2-(4-tert-butylphenoxymethyl)-5-(2-phenylazetidine-1-carbonyl)pyrimidin-4-ol
3-(propan-2-yl)-5-[1-(thiophene-3-sulfonyl)pyrrolidin-2-yl]-1,2,4-oxadiazole
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[(2-phenylpropyl)amino]piperidin-1-yl}benzamide
2-chloro-3-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
2-ethyl-N-[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]pyrimidine-5-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1,3-benzoxazole
6-methoxy-2-oxo-N-[2-(pyrazin-2-yl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-{1-[1-(4-methoxyphenyl)piperidin-4-yl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
2-fluoro-6-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
ethyl 4-[(3-fluorophenyl)methyl]-1-[2-(5-oxopyrrolidin-2-yl)acetyl]piperidine-4-carboxylate
6-cyano-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}pyridine-3-carboxamide
4-{2-phenyl-2-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}phenol
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-4,4,4-trifluorobutan-1-one
ethyl 4-[({2-[3-(dimethylamino)-2-hydroxypropoxy]-5-methoxyphenyl}methyl)amino]piperidine-1-carboxylate
(3R,5R)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-[2-(dimethylamino)ethyl]-9-[(1R,2S)-2-propylcyclopropanecarbonyl]-2,9-diazaspiro[5.5]undecan-3-one
N,N-diethyl-1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)pyrrolidin-3-amine
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(2-methylpyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-({5-[1-(3-fluorophenyl)-1H-pyrazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
N-(3-fluorophenyl)-6-[4-(furan-2-yl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
6-methyl-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one