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2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
1-[(2-chlorophenyl)methyl]-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(2-methoxyethyl)-6-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]-1,3-benzoxazole
5-ethyl-4-[4-(pyrazin-2-yl)piperazin-1-yl]pyrimidin-2-amine
1-[1,3-dioxo-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-(2,2-diphenylethyl)piperidine-3-carboxamide
2-[3-oxo-3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
1-(3-chlorothiophene-2-carbonyl)-4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}pyridazine-3-carboxamide
1-(1-benzoxepine-4-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-{[2-(2-fluorophenyl)ethyl]amino}-5-methyl-N-[2-(pyridin-4-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-2-yl)pyridine
(2S,4R)-N-methyl-4-{[(3-phenoxyphenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-ethyl-4-(methoxymethyl)-5-methyl-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-[2-(dimethylamino)ethyl]-N-methyl-1-[(8-methylquinolin-5-yl)methyl]piperidin-4-amine
N-({7-[(2-chloro-3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
2,3,5-trimethyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
N4-(1-benzothiophen-5-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}pent-4-enamide
N-[(2R,3R)-1'-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-(6-ethylpyridin-2-yl)-5-[1-(2-methoxyacetyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1-{5-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
2-(2-chloro-4-fluorophenyl)-1-{3-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}ethan-1-one
N-(1-methyl-1H-pyrazol-3-yl)-2-{4-[1-(4-methylpyridin-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}acetamide
3-phenyl-N-{1-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-methyl-2-(1-methyl-1H-pyrrole-2-carbonyl)-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N,4-dimethyl-2-(methylamino)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1,3-thiazole-5-carboxamide
3-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,9-diazaspiro[5.5]undecane
5-[4-hydroxy-1-(2-methylbutyl)piperidin-4-yl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1-benzofuran-2-carboxamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
[(2,4-difluoro-3-methoxyphenyl)methyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
2-chloro-N-({1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]piperidin-3-yl}methyl)benzamide
1-ethyl-N-[2-(4-fluorophenyl)-2-hydroxyethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-[(2,3-dimethoxyphenyl)methyl]-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
({1-[1-(2,2-diethylcyclopropanecarbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)dimethylamine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(dicyclopropylmethyl)-N-methylpiperidine-3-carboxamide
4-(1-cyclopentanecarbonylpiperidin-4-yl)-5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidine
N-(2,6-dimethylphenyl)-3-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]benzamide
N-cyclopentyl-3-{[1-(pyrimidin-4-yl)ethyl]sulfamoyl}benzamide
5-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}pyrimidin-2-amine
5-(4-methyl-1H-imidazol-5-yl)-1-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-4-phenyl-1H-imidazole
3,4-difluoro-N-[(3-methylpyridin-4-yl)methyl]benzamide
2-butyl-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-1,3-benzoxazole-5-carboxamide
N-[(4-fluorophenyl)methyl]-5-methyl-1-propyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
5-{2-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-[2-(2-oxopiperidin-1-yl)ethyl]benzamide
N-{2-[(1,3-thiazol-2-yl)carbamoyl]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-{4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
1-cyclohexyl-3-hydroxy-4-(quinolin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one