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1-(2-methylphenyl)-3-{1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
(4aS,8aS)-2-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-decahydroisoquinolin-4a-ol
2-{1-[(2-ethoxyphenyl)methyl]-4-(pyridine-3-carbonyl)piperazin-2-yl}ethan-1-ol
6-phenyl-3-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-[4-({2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}methyl)phenyl]acetamide
4-{[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]amino}butan-1-ol
4-(6-aminopyridine-3-carbonyl)-1-(3-methoxyphenyl)piperazin-2-one
(5S,9aS,9bS)-5-(1-benzofuran-2-yl)-2-[(3-chlorophenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-(prop-2-en-1-yl)propanamide
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-(3-methoxyphenyl)-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazin-2-one
3-methyl-5-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrazole
methyl 4-[2-amino-3-cyano-6-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyridin-4-yl]-1H-pyrazole-3-carboxylate
5-methoxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyrimidin-2-amine
(2S,4S)-4-amino-N-methyl-1-[4-(4-propylphenyl)benzoyl]pyrrolidine-2-carboxamide
4-(3-ethyl-1H-pyrazole-4-carbonyl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
[(2S,6S)-4-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-(1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)piperidin-3-ol
N-methyl-4-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-thiazol-2-amine
N-ethyl-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-(2-methylprop-2-en-1-yl)piperidine-4-carboxamide
2-[5-(1,1-dioxo-1λ6-thiolan-3-yl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
N,4,6-trimethyl-2-oxo-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]amine
(2R,3R)-1'-[(5-ethylfuran-2-yl)methyl]-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
methyl 4-{[(2-{5-oxo-1-[2-(thiophen-2-yl)ethyl]pyrrolidin-2-yl}ethyl)amino]methyl}benzoate
[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})amine
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(1-methyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(5-{[(2,5-dimethylphenyl)methyl]amino}-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-ol
7-(cyclobutylmethyl)-2-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
5-({4-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-1,3-oxazol-2-yl}methoxy)isoquinoline
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-(2-methylphenyl)-1,2,4-triazin-3-amine
methyl 4-({[(3R,5S)-1-benzyl-5-(methylcarbamoyl)pyrrolidin-3-yl]amino}methyl)benzoate
4-{5-[(2S)-1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
N-[2-(3,4-dimethoxyphenyl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-(6-fluoro-4-methylquinazolin-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)piperidin-4-amine
(5S,9aS,9bS)-2-cyclopentyl-5-(4-ethynylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3S,4R)-4-(3-fluorophenyl)-1-(6-methoxyhexanoyl)pyrrolidine-3-carboxylic acid
3-{1-[(4-phenylphenyl)methyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
(1R,5R)-6-[4-(1H-imidazol-1-yl)butanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-[1-(2,2-dimethylpropyl)-4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl]ethan-1-ol
2-methyl-4-[1-(oxolan-3-ylmethyl)piperidin-4-yl]pyrimidine
7-{[4-(2-methoxyethoxy)phenyl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
4-methoxy-2-methyl-N-[2-(1-methylpiperidin-3-yl)ethyl]benzamide
2-ethyl-5-{[1,2,4]triazolo[4,3-c]quinazolin-3-yl}pyrimidine
2-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
2-(adamantan-1-yl)-N-[2-(dimethylamino)ethyl]-N-ethyl-4-hydroxypyrimidine-5-carboxamide
N-({3-[3-(benzyloxy)propyl]phenyl}methyl)acetamide
8-(1H-1,3-benzodiazol-2-ylmethyl)-1-ethyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
{1-[(2-cyclohexylpyrimidin-5-yl)methyl]azepan-2-yl}methanol