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2-(3-fluoro-4-hydroxyphenyl)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]ethan-1-one
2-[4-(5-{[(2-methoxyphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]-2-oxoacetamide
1-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
9-(cyclopropylmethyl)-1-methyl-4-(1-methyl-1H-pyrazole-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
9-(4,6-dimethylpyrimidin-2-yl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(3-hydroxy-3-methylbutyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]benzamide
3-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-1,2-dimethyl-1H-indol-5-ol
(1-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)(thiophen-2-yl)methanol
4-ethyl-6-[4-({imidazo[1,2-a]pyridin-3-ylmethyl}amino)piperidin-1-yl]-N,N-dimethylpyrimidin-2-amine
1-tert-butyl-4-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}pyrrolidin-2-one
1-ethyl-2-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,2-dihydropyridine-4-carboxamide
2-[4-(methylsulfanyl)phenyl]-1-[3-(morpholine-4-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chlorophenyl)urea
1-{3-[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]propyl}pyrrolidin-2-one
methyl({[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
2-(4-{[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
N-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-10-azabicyclo[4.3.1]decane-10-carboxamide
ethyl 1-(3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanoyl)piperidine-3-carboxylate
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-[2-(2-methoxyphenyl)ethyl]-2-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}quinazolin-4-amine
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-6-methylimidazo[1,2-a]pyridine-2-carboxamide
1-[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethane-1,2-dione
[(3R,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
(2S)-2-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]formamido}-3,3-dimethylbutanoic acid
9-[(2R)-2-amino-3-methoxypropanoyl]-2-(furan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
methyl 2-(2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamido)acetate
(1R,9aR)-1-[({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
3-[4-(2,3,5,6-tetramethylbenzoyl)piperazin-1-yl]pyrazine-2-carbonitrile
1-[2-(morpholin-4-yl)ethyl]-3-[6-(trifluoromethyl)pyridin-3-yl]urea
7-(cyclobutylmethyl)-2-(5-ethyl-1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
1-(2,6-dimethylpyridin-4-yl)-4-(4-ethyl-5-methylthiophene-3-carbonyl)piperazine
2-[4-chloro-2-({3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)phenoxy]acetic acid
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-methyl-N-propylacetamide
N-[2-(dimethylamino)ethyl]-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
ethyl[(4-methoxy-2-methylphenyl)methyl][(1-methyl-1H-imidazol-2-yl)methyl]amine
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
N-[(3R,4S)-1-(2-carbamoylethyl)-4-cyclopropylpyrrolidin-3-yl]-1,2,3,4-tetrahydroquinoline-8-carboxamide
3-{5-[(4-methyl-1H-pyrazol-1-yl)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
[(2E)-3-(furan-2-yl)prop-2-en-1-yl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
3-[(2,6-difluorophenyl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-cyclopropyl-3-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
6-[3-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-oxopropyl]-2,3-dihydropyridazin-3-one
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-4-(4-fluorophenyl)butane-1,4-dione
(2R,3R)-3-{[(5-ethylpyridin-2-yl)methyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol