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1-(1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)piperidin-3-ol
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-propyl-1,3-thiazole
2-[2-fluoro-6-(propan-2-yloxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-{[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}-4-methoxyphenol
8-(5-ethyl-2-methylpyrimidin-4-yl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
5-{[ethyl(2,2,2-trifluoroethyl)carbamoyl]amino}-N,N-dimethyl-1-benzothiophene-2-carboxamide
ethyl 4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
methyl 3-(3-methylbutanoyl)-7-oxo-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-({4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
2-(2H-1,2,3-benzotriazol-2-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
2-{[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methylpyrazine-2-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
1-[3-({2-[(3-fluorophenyl)methyl]morpholin-4-yl}methyl)phenyl]ethan-1-one
1-{7-methylthieno[3,2-d]pyrimidin-4-yl}-N-[3-(pyridin-4-yl)propyl]piperidin-4-amine
N4,5,6-trimethyl-N4-[(4-methyl-1,3-thiazol-2-yl)methyl]pyrimidine-2,4-diamine
4-{1-[1-(4-methylpyrimidin-2-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
2-benzyl-8-(pyrazine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(3S,5S)-1-benzyl-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-[(2,5-dimethylphenyl)methyl]pyrrolidin-3-amine
N,2-dimethyl-N-{2-phenyl-1-[1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]ethyl}furan-3-carboxamide
[(1-methyl-1H-pyrazol-4-yl)methyl]({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl})(propan-2-yl)amine
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-2-(thiophen-2-yl)azetidine
2-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]-3-(furan-2-yl)propanoic acid
1-(azepan-1-yl)-3-(3-{[methyl(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
4-benzyl-3-ethyl-1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-1,4-diazepan-5-one
2-methyl-N-(2-{[(4-methylphenyl)methyl]sulfanyl}phenyl)-5-oxo-1,4-diazepane-1-carboxamide
N,2-dimethyl-N-(1,2-oxazol-5-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-phenoxyethan-1-one
1-[(3-fluorophenyl)methyl]-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
1-[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
(3R,4R)-1-(4-chloro-1H-pyrazole-3-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1,3,7-trimethyl-2-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1H-indole
1-(2,3-dihydro-1H-inden-2-yl)-4-({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amino)pyrrolidin-2-one
4-(4-chlorophenyl)-1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-ol
N,N-dimethyl-6-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyridine-3-carboxamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(1H-imidazol-1-yl)benzamide
2-[1-(3-methylbutyl)-4-(1H-pyrazol-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-({1-[(5-chloro-2,3-dimethoxyphenyl)methyl]pyrrolidin-3-yl}methyl)acetamide
N-[2-(3-methoxyphenyl)phenyl]-1-{[3-(methylsulfanyl)phenyl]methyl}piperidine-4-carboxamide
2-(4-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenyl)ethan-1-amine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(pyrimidin-2-ylsulfanyl)acetamide
7-fluoro-3-({methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
ethyl 4-{[(1R,2S)-2-[2-(1H-indol-3-yl)acetamido]cyclobutyl]amino}piperidine-1-carboxylate
N-benzyl-2-({[(1-ethyl-1H-imidazol-2-yl)methyl]amino}methyl)-N-methyl-2,3-dihydro-1H-inden-2-amine
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2,8-dimethylquinoline-4-carboxamide
N-[2-(2-chloro-6-fluorophenyl)ethyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
5-[(2-fluorophenyl)methyl]-5-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
4,6,7-trimethyl-2-[4-(thiophen-3-ylmethyl)-1,4-diazepan-1-yl]quinazoline
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
[(2S,6S)-4-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol