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N-({3-methyl-7-[(2E)-3-phenylprop-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(pyrimidin-2-ylsulfanyl)acetamide
N4-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-5,6-dimethylpyrimidine-2,4-diamine
(3S,7S)-5-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-methoxy-3-[2-(4-methoxy-2,5-dimethylphenyl)-1H-imidazol-1-yl]pyridine
7-fluoro-N,2-dimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]quinoline-4-carboxamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(N-phenylmethanesulfonamido)propanamide
8-methyl-2-propyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
2-{4-[(6-chloroquinolin-2-yl)methyl]-1-(2,2-dimethylpropyl)piperazin-2-yl}ethan-1-ol
2-{5-[5-(2-chlorophenyl)furan-2-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
1-[(2-fluorophenyl)methoxy]-8-[1-(2-methylpropyl)-5-oxopyrrolidine-3-carbonyl]-1,8-diazaspiro[4.5]decan-2-one
2-[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]pyridine-3-carboxamide
N-[(2R,3R)-1'-(dimethyl-1,3-thiazole-5-carbonyl)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}-1,4-dihydropyridine-3-carboxamide
2-(2,4-dimethylphenyl)-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid
5-amino-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1H-pyrazole-3-carboxamide
4-(4-{[(2-methoxyphenyl)methyl]amino}piperidin-1-yl)-N-(1-phenylethyl)benzamide
3-(1-methanesulfonylpiperidin-4-yl)-1-[2-(5-methylfuran-2-yl)phenyl]urea
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)pent-4-enamide
4-ethyl-1-methyl-3-{1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-4-(pyridin-4-yl)-1-(quinoxalin-2-yl)pyrrolidine-3-carboxylic acid
1-(2-methoxyquinoline-4-carbonyl)-N,N-dimethylazepan-4-amine
N-[3-(dimethylamino)-1-phenylpropyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[(3-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}-4-methoxyphenyl)methyl]piperidine-4-carboxamide
4-[2-(2-ethoxyphenyl)acetyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-{[(1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
2-[2-(3-fluorophenyl)piperidine-1-carbonyl]-6-methyl-4H-pyran-4-one
1-{[2-chloro-6-methoxy-4-(2-methoxyphenoxy)phenyl]methyl}pyrrolidine
3-(but-2-yn-1-yl)-5-(2-phenylethyl)-5-[1-(quinolin-5-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
2-(4-chlorophenoxy)-N-{2-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}acetamide
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-(pyrazine-2-carbonyl)-1,4-diazepane
2-(butylsulfanyl)-N4-(oxan-2-ylmethyl)pyrimidine-4,6-diamine
4-(5-acetylthiophene-3-carbonyl)-1-benzyl-6-(cyclopropylmethoxy)-1,4-diazepan-2-one
N-[(3-fluoro-4-methylphenyl)methyl]-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
3-[2-chloro-5-(morpholin-4-yl)phenyl]-1-methyl-1-[1-(pyridin-2-yl)ethyl]urea
1-[9-(2,3-dihydro-1H-inden-1-yloxy)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
6-[3-oxo-3-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propyl]-2,3,4,5-tetrahydropyridazin-3-one
5-methyl-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N5,N5,N6-trimethyl-N6-(pyrazin-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-benzyl-3-{[(2-hydroxypropyl)amino]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
2,5-dimethyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}thiophene-3-sulfonamide
N-[(3,4-dimethoxyphenyl)methyl]-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
N-methyl-4-(piperidin-1-ylmethyl)-N-(prop-2-en-1-yl)benzamide
N-(1-{7-[(2-chloro-4,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylfuran-3-carboxamide
(4aS,7aR)-1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-fluoro-2-(4-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}piperazin-1-yl)pyrimidine
1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-(oxolan-2-ylmethyl)piperazine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-3-(pyridin-4-yl)propanamide
3-(2-methyl-1H-indol-1-yl)-N-[3-(3-oxopiperazin-1-yl)propyl]propanamide
methyl 3-{[5-(2-chlorophenyl)furan-2-yl]methyl}-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate