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3,5-dichloro-N-(2-hydroxyethyl)-4-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl){[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amine
5-ethyl-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrimidin-2-amine
N-{1-[1-(4-fluorobenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylthiophene-3-carboxamide
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-4-phenylbutane-1,4-dione
3-[5-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-3-yl)-1,2,4-oxadiazol-3-yl]pyridine
7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-4-[(2E)-2-methylbut-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(2-methoxyacetyl)-N-[3-(pyridin-3-yl)phenyl]-1,4-diazepane-1-carboxamide
6-(2-chlorophenyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-(pyrazin-2-ylmethyl)-1H-pyrazole-3-carboxamide
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl){[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}amine
N-methyl-2-(3-methylpentanamido)-7-oxo-N-(propan-2-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
(3S,4R)-1-(1-benzylpiperidin-4-yl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
3,5-dimethyl-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-indole-2-carboxamide
6-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]pyrrolidin-3-yl}piperidine
N-(2-ethylphenyl)-3-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]propanamide
1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-3-(1H-imidazol-1-ylmethyl)piperidine
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-(thiophen-3-yl)propan-1-one
N-{2-methoxy-4-[2-(1H-1,2,4-triazol-1-yl)propanamido]phenyl}-2,2-dimethylpropanamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]-N-methylpiperidine-3-carboxamide
2-(4-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)phenol
benzyl(1H-imidazol-2-ylmethyl)[(4-methyl-1,3-thiazol-5-yl)methyl]amine
N-{[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
3-{4-[({[4-(hydroxymethyl)phenyl]methyl}carbamoyl)amino]phenyl}-N,N-dimethylpropanamide
N-methyl-3-[1-(9H-purin-6-yl)piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-{4-[(8-chloro-4-hydroxyquinolin-2-yl)methyl]piperazin-1-yl}-N-(propan-2-yl)acetamide
5-({[(3-{2-[4-(2,2-diphenylacetyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
(2R,3S,6R)-3-phenyl-5-(4,4,4-trifluorobutyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(3-methoxypropyl)-6-{octahydropyrrolo[1,2-a]piperazin-2-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-chloro-N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1H-indole-2-carboxamide
1-[(4-fluorophenyl)methyl]-N-(1-hydroxy-2-methylpropan-2-yl)-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-1-(2-methoxyphenyl)piperidin-4-amine
2-(2-methyl-4-{[2-(piperidin-1-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)acetic acid
3-methyl-1-{1-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]piperidin-4-yl}butan-1-ol
5-(2,6-dichlorophenoxymethyl)-3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazole
N-[2-(1H-pyrazol-4-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
{1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
2-[4-(2-methoxybenzoyl)piperazin-1-yl]-4-(pyridin-2-yl)pyrimidine
9-(2,5-dimethylfuran-3-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
(1S,5R)-6-methyl-3-(3-phenoxypropanoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3aS,6aR)-5-[(3,4-difluorophenyl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(2-methoxyethyl)methylamine
3-{imidazo[1,2-a]pyridin-2-ylmethyl}-8-methoxy-3,4-dihydroquinazolin-4-one
3-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenol
N-[3-(cyclohexylsulfanyl)propyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide