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N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetamide
4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
3-{[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
2-(2,3-dihydro-1H-inden-5-yloxy)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-methylpropan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[(2S)-2-carbamoylpyrrolidin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-ethyl-1-[2-(piperidin-2-yl)ethyl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-(6-methoxypyridin-3-yl)thiophene-2-carboxamide
2-chloro-4-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}phenol
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-2-carboxamide
5-methyl-3-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-2,3-dihydro-1,3-benzoxazol-2-one
2-{[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-N-cyclopropylacetamide
2-(4-methylnaphthalen-1-yl)pyridine-4-carboxamide
methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)[(3-methylquinoxalin-2-yl)methyl]amine
1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-methoxypiperidine
2-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-1-methyl-1H-1,3-benzodiazole
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-butyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1-(3-methylcinnolin-5-yl)urea
6-({2-[ethyl(methyl)amino]-2-methylpropyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
methyl 3-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
3-amino-N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
2-(4-acetylpiperazin-1-yl)-2-(4-fluoro-2-methoxyphenyl)acetic acid
ethyl 4-[(4-chlorophenyl)methyl]-1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidine-4-carboxylate
3-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-phenoxyphenyl)urea
N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-4-(trifluoromethyl)benzamide
(1S,5R)-3-[(2-aminopyridin-3-yl)methyl]-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({1-[(2,5-dimethylphenyl)methyl]piperidin-3-yl}methyl)-4-fluorobenzamide
3-methyl-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1,2-dihydroquinoxalin-2-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[1-(propan-2-yl)piperidin-4-yl]pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
1-[benzyl(methyl)amino]-3-(4-{[(2-methoxyethyl)(propan-2-yl)amino]methyl}phenoxy)propan-2-ol
N'-{[4-methoxy-3-(oxolan-3-ylmethoxy)phenyl]methyl}-N,N-dimethyl-N'-(pyridin-3-ylmethyl)butanediamide
N-benzyl-N-ethyl-3,5-dimethyl-1-benzofuran-2-carboxamide
2-(3-fluorophenoxymethyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
2,6-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)quinoline-3-carboxamide
N,1,3-trimethyl-N-{2-phenyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]ethyl}-1H-pyrazole-5-carboxamide
2-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-cyclobutanecarbonyl-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4-diazepane
(1R,5R)-6-(cyclobutylmethyl)-3-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-methyl-1H-1,2,3-benzotriazole-5-carboxamide
4-(1H-pyrazol-1-yl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidine-4-carboxylic acid
N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-indole-6-carboxamide
(2-{2-[1-(1H-1,2,3-benzotriazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N,N-diethyl-1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
2-(adamantan-1-ylsulfanyl)-N-(1H-imidazol-2-ylmethyl)-N-methylacetamide
2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,4-dihydroquinolin-4-one
2,4-dimethyl-N-[4-(4-{[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}piperidin-1-yl)phenyl]benzamide
1-(benzyloxy)-8-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-1,8-diazaspiro[4.5]decan-2-one