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2-cyclohexyl-5-{1-[(1-ethylpyrrolidin-2-yl)methyl]-1H-imidazol-2-yl}pyrimidine
(3S,5R)-1-(2-phenylethyl)-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
4-[4-methyl-5-(morpholine-4-carbonyl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
N-[(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)methyl]-3-phenylpropanamide
1-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(oxan-2-ylmethyl)piperidine-4-carboxylic acid
4-[(2,2-dimethylpropyl)amino]-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
1-(2-cyclopentyl-2-phenylethyl)-3-(2-hydroxypyridin-3-yl)urea
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(piperidin-3-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(3-methylphenyl)ethan-1-one
5-cyano-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
3-benzyl-N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
2-(4-{[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]amino}piperidin-1-yl)pyridine-4-carbonitrile
4-ethyl-1-[2-(1-methylpiperidin-2-yl)ethyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N,N-diethyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
(3R)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3,4,4-trimethylpyrrolidin-3-ol
9-(propane-1-sulfonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 5-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{4-[(3-methoxypiperidin-1-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
1-{3-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-methoxyethan-1-one
N-{4-[1-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1H-1,2,3-triazol-4-yl]phenyl}acetamide
N'-[(1S)-2-hydroxy-1-phenylethyl]-N-[2-(methylsulfanyl)phenyl]butanediamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(pyridin-3-yl)ethane-1,2-dione
2-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxo-N-(propan-2-yl)acetamide
1-{3-[4-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}methyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
6-(dimethyl-1,2-oxazol-4-yl)-N-propylpyridine-3-carboxamide
6-(2,5-dimethylphenyl)-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[3-(propan-2-yloxy)propyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
(1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-(trifluoromethyl)benzamide
N-[2-(2,5-dimethylphenoxy)ethyl]-N-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
2-(1-cyclohexylpiperidin-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}acetamide
2-(1,2-benzoxazol-3-yl)-N-{1-oxaspiro[4.4]nonan-3-yl}acetamide
9-[1-(2-fluorophenyl)cyclopropanecarbonyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(2-methoxyethyl)-2-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-1-(propan-2-yl)piperidine-3-carboxamide
2-(3-hydroxyphenyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
4-(5-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1,3-benzothiazole-6-carboxamide
9-[5-(methoxymethyl)thiophene-2-carbonyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-N-(2-methylpropyl)-6-oxo-N-(3-phenylprop-2-yn-1-yl)-1,6-dihydropyrimidine-5-carboxamide
2-{2-[1-(8-fluoroquinoline-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
1-{2-[(6-methyl-2-propylpyrimidin-4-yl)amino]ethyl}piperidin-4-ol
1-(2-methoxyphenyl)-N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]oxy}benzamide
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
7-(2,6-dimethoxyphenyl)-9-methoxy-4-(propan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-benzyl-3-(1-benzylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one