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1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-2-(furan-2-yl)azepane
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-ol
N-{1-[1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidin-4-yl]pyrrolidin-3-yl}acetamide
1-(pyridin-3-ylmethyl)-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yloxy)ethyl]acetamide
N-{2-[(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazol-4-yl)formamido]ethyl}acetamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,5-dimethylfuran-2-carboxamide
(3S,4S)-4-cyclopropyl-1-{2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}pyrrolidine-3-carboxylic acid
7-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-[1-(propan-2-yl)-4-[(2,4,5-trimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
8-(3-methylthiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,4-dihydroquinolin-4-one
8-(1-hydroxypropan-2-yl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(4-chlorobenzenesulfonamido)ethyl]-5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
1-{4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3-cyclohexylpropan-1-one
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
1-(4-methyl-1H-pyrrole-2-carbonyl)-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
(3S,5S)-5-[(pyridin-4-ylmethyl)carbamoyl]-1-[(1r,4r)-4-methylcyclohexanecarbonyl]piperidine-3-carboxylic acid
3,6-dimethyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}[1-(pyridin-4-yl)propyl]amine
3-cyclopropyl-5-[6-methyl-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridin-4-yl]-1H-1,2,4-triazole
5-[4-(2-fluorophenoxy)piperidine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
5-fluoro-2-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H-1,3-benzodiazole
4-oxo-N-(oxolan-3-yl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]-2-phenylethane-1,2-dione
2-(5-acetylthiophen-3-yl)-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}acetamide
N-[2-({2-[(quinolin-6-yloxy)methyl]-1,3-oxazol-4-yl}formamido)ethyl]acetamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[(3R,4S)-4-cyclopropyl-1-(2,5-dimethylfuran-3-carbonyl)pyrrolidin-3-yl]acetamide
2-[1-(2,6-dimethylpyridine-4-carbonyl)piperidin-2-yl]ethan-1-ol
1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-[(dimethylamino)methyl]piperidin-3-ol
4-methyl-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-[2-(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclobutanecarboxamide
4-(4-ethoxy-3-methylphenyl)-4-oxo-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]butanamide
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-4-[2-(pyrrolidin-1-yl)ethyl]piperazine
6-[(3-hydroxyphenyl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
4-[4-(ethanesulfonyl)piperazin-1-yl]-6-(piperidin-3-yl)pyrimidine
N-[2-(1H-imidazol-4-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
4-ethenyl-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)benzamide
3-methoxy-N-{1-methyl-2-phenyl-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-7-yl}propanamide
4-[2-(4-methoxyphenyl)ethyl]-4-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
6-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
4-[3-(propan-2-yl)-1H-pyrazol-1-yl]-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxylic acid
N-[2-(3-fluorophenyl)ethyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
1-(2-cyclohexylethyl)-3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-3-hydroxypiperidin-2-one
4-(hydroxymethyl)-1-(2-methoxypyridine-4-carbonyl)piperidin-4-ol
N-cyclopropyl-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
1-[(3-{[1-(furan-3-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}isoquinoline