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9-(2-acetylbenzoyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-ethoxyphenyl)piperazine
N-cyclooctyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propanamide
1-[2-({[2-(methylsulfanyl)phenyl]carbamoyl}amino)ethyl]piperidine-3-carboxamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-4,6-dimethyl-2-oxo-2H-pyran-5-carboxamide
2-(6-methoxypyridin-3-yl)-2-[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amino]acetic acid
4-({1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
N-(2,3-dihydro-1H-inden-1-yl)-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
methyl 2-(benzylsulfamoyl)-6-[(2-methoxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-methanesulfonyl-1'-(2-phenylethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-chloro-3-{[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]methyl}-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
2-[(3-fluorophenyl)methyl]-4-{4-[3-(hydroxymethyl)piperidine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[(3R,4S)-1-acetyl-4-(propan-2-yl)pyrrolidin-3-yl]-5-(propan-2-yl)thiophene-3-carboxamide
1-(propan-2-yl)-N-[4-(pyridin-2-yl)butyl]-1H-pyrazole-4-carboxamide
1,3-dimethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-({7-[(2-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
4-(5-aminopyrazin-2-yl)-N-tert-butylbenzene-1-sulfonamide
3-benzyl-4-[(4-hydroxy-6-methylquinolin-2-yl)methyl]piperazin-2-one
N-[2-(2,3-dichlorophenyl)ethyl]-4-(1H-pyrazol-4-yl)butanamide
N-({5-[(2-fluoro-5-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
4-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methoxypyrimidine
(1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanol
[(3,4-difluorophenyl)methyl](methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
N-({1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
4-(1H-1,2,3,4-tetrazol-1-ylmethyl)-N-[1-(thiophen-2-yl)propan-2-yl]benzamide
N-[(2-chlorophenyl)methyl]-4-cyano-N-(2-methoxyethyl)-1H-pyrrole-2-carboxamide
N-[2-(4-chlorophenyl)ethyl]-2-{methyl[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amino}acetamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]acetamide
(2R,4S)-1-[(2-chloro-6-fluorophenyl)methyl]-4-hydroxypiperidine-2-carboxylic acid
4-[2-(benzyloxy)acetyl]morpholine-2-carboxylic acid
2-(6-cyclopropylpyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
5-{1-[2-(2-chloro-6-fluorophenyl)acetyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
8-{3-[4-(3-methylphenyl)piperazin-1-yl]propanoyl}-2,8-diazaspiro[4.5]decan-3-one
methyl[(1-methyl-1H-indol-3-yl)methyl][(3-methylpyridin-4-yl)methyl]amine
(3R,4S)-4-cyclopropyl-1-(5-methyl-1H-indazole-3-carbonyl)pyrrolidin-3-amine
1-{2-methoxy-4-[(4-methylpiperidin-1-yl)methyl]phenoxy}-3-(morpholin-4-yl)propan-2-ol
6-{2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-imidazol-1-yl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-amino-6-[4-(4-cyclobutyl-6-methylpyrimidin-2-yl)piperazin-1-yl]-3,4-dihydropyrimidin-4-one
N-(pyridin-2-ylmethyl)-4-[4-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(4-hydroxypiperidin-1-yl)-N-propyl-N-(thiophen-3-ylmethyl)acetamide
N-(6-methoxyquinolin-8-yl)-4-(2-oxo-1,3-oxazolidin-3-yl)piperidine-1-carboxamide
(5-{1-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-imidazol-2-yl}furan-2-yl)methanol
7-(2-propoxybenzoyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(4-{[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}piperazin-1-yl)-1-(pyrrolidin-1-yl)ethan-1-one
1-{5-methoxy-2-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]phenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
2-[(1-acetylpiperidin-4-yl)oxy]-N-benzyl-5-chloro-N-(2-hydroxyethyl)benzamide
N-[2-(1-{[5-chloro-2-(trifluoromethyl)phenyl]methyl}piperidin-2-yl)ethyl]acetamide
5-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione