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2-[5-(5-acetylthiophen-2-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]acetamide
3-(diphenylmethyl)-5-(oxane-4-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-ethyl-4-methyl-2-(pyridin-3-yl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
8-[(2-chloro-3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
2,6,8-trimethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]quinoline-4-carboxamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3,6,7-trimethyl-1-benzofuran-2-carboxamide
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-3-methoxypyridine-2-carboxamide
N-[(3-methoxyphenyl)methyl]-3-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]propanamide
1-{1-[1-(4,6-dimethylquinazolin-2-yl)piperidine-4-carbonyl]piperidin-4-yl}-2-phenylethan-1-ol
2-{2-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
1-[2-(1H-imidazol-1-yl)ethyl]-4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
1-[5-(4-chloro-3,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)-N-methylacetamide
[(2S)-1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
6-methyl-1-(2-methylphenyl)-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperazin-2-one
N-[(2-amino-1,3-thiazol-4-yl)methyl]-1-(3,4-difluorophenyl)-5-oxopyrrolidine-3-carboxamide
8-(furan-2-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(furan-2-ylmethyl)-5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
N-{[7-(1-benzofuran-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-oxopyrrolidine-3-carboxylic acid
6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyridazin-3-amine
benzyl(1H-imidazol-2-ylmethyl)(1,3-thiazol-2-ylmethyl)amine
2-{5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}pyridine
1-[2-(dimethylamino)ethyl]-3-{2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl}-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
2-[4-(1,2-oxazol-3-ylmethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
2-(2-methoxyethyl)-8-(pyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
4-[1-(3,4-dimethylbenzoyl)piperidin-3-yl]-2-methyl-5-(3-methylphenyl)pyrimidine
2-[8-(1,3-benzothiazol-2-ylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
1-(5-chloronaphthalene-1-carbonyl)-4-cyclobutanecarbonyl-1,4-diazepane
N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-1H-pyrrole-2-carboxamide
1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-{5-[(3-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}urea
4-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-1,4-oxazepan-6-ol
2-(dimethylamino)-N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-4-methylpyrimidine-5-carboxamide
N-cyclopropyl-3-{1-[4-(morpholin-4-yl)benzoyl]piperidin-3-yl}propanamide
2-(2-{[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}ethyl)-6-methyl-3,4-dihydropyrimidin-4-one
1-[4-({benzyl[(4-methyl-1,3-thiazol-5-yl)methyl]amino}methyl)thiophen-2-yl]ethan-1-one
4-(4-benzyl-1H-pyrazol-5-yl)-1-(furan-3-ylmethyl)piperidine
1-(5-chloro-2-methylphenyl)-4-(1-cycloheptyl-1H-1,2,3-triazole-4-carbonyl)piperazine
2-[(3-methoxyphenyl)amino]-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)butanamide
1-(4-{4-[(3R)-3-hydroxypyrrolidine-1-carbonyl]phenoxy}piperidin-1-yl)-3-methoxypropan-1-one
N-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-N,2,2-trimethyloxan-4-amine
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide
5-(methoxymethyl)-N-({7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)furan-2-carboxamide
N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl 3-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
7-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-(2-hydroxy-2-phenylethyl)-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methylbenzamide
1-(4-{[4-(dimethylamino)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2-phenylethan-1-ol