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ethyl 1-[3-(1,2-oxazinan-2-yl)propanoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
1-({3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}sulfonyl)azepane
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(4-methoxyphenyl)methyl]propanamide
4-{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}-1,3-dimethylpiperazin-2-one
4-(2-methylpropyl)-1-[2-(2,3,4-trifluorophenyl)acetyl]-1,4-diazepan-5-one
3-[5-(1,2,5-thiadiazole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-oxo-2,3,4,5-tetrahydro-1,5-benzothiazepine-7-sulfonamide
9-(5-methoxyfuran-2-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1-ethyl-5-oxopyrrolidin-3-yl)-4-(1H-1,2,4-triazol-1-yl)butanamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(2-methoxypyridine-3-carbonyl)-N-methylpiperidin-3-amine
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methylacetamide
N-[(3R,4R)-1-[(5-ethylpyridin-2-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
(2-ethoxy-5-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}phenyl)methanol
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-7-(2-chlorobenzamido)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
(1-benzothiophen-2-ylmethyl)(methyl){[4-({1-[2-(trifluoromethyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}amine
2-chloro-9-methyl-3-{[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amino]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
1,3-dimethyl-6-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(8-hydroxyquinolin-2-yl)-1-methyl-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-phenyl-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]pyrimidin-2-amine
1-({2-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)azetidin-3-ol
2-(4-fluorophenyl)-N,N-dimethylpiperidine-1-sulfonamide
(2S,4R)-N-[2-(2-fluorophenyl)ethyl]-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)hexan-1-one
4-(furan-3-ylmethyl)-3-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)piperazin-2-one
N-{1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}thian-4-amine
N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
2-(1-methylpyrrolidin-3-yl)-9-(2-propoxyacetyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[furan-2-yl(phenyl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl)ethan-1-ol
5-(1,6-dimethyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
2-methyl-5-[2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
{3-[(4-fluorophenyl)methyl]-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl}methanol
4-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-1-(4-methoxyphenyl)piperazin-2-one
3,5-dimethyl-4-{2-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]ethyl}-1,2-oxazole
(3S,5R)-1-(4-ethylbenzoyl)-5-(4-methylpiperazine-1-carbonyl)piperidine-3-carboxylic acid
7-[(3-chloro-1H-indol-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-acetamido-N-[4-(pyridin-2-ylmethoxy)phenyl]pyrrolidine-1-carboxamide
1-cyclobutanecarbonyl-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-1,4-diazepane
N-cyclopentyl-4-fluoro-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzene-1-sulfonamide
3-methyl-5-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridin-2-amine
5-(furan-2-yl)-1-(1-phenylethyl)-1H,4H-pyrazolo[3,4-d]imidazole
6-[3-(morpholin-4-ylmethyl)phenyl]-N-(propan-2-yl)pyrimidin-4-amine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-5-(naphthalen-2-yl)-1,2,4-triazin-3-amine
3-(3-methoxyphenyl)-N-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
5-[(2-chlorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(2-methylbenzoyl)piperidin-4-yl]imidazolidine-2,4-dione
7-[(2S)-2-amino-3,3-dimethylbutanoyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-methoxy-4-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}phenol