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ethyl 4-oxo-5-phenoxy-1-[1-(1H-pyrazol-1-yl)propan-2-yl]-1,4-dihydropyridine-3-carboxylate
3-(cyclobutylsulfamoyl)-N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
5-cyclobutanecarbonyl-1'-(3-methyloxetane-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
{4-benzyl-1-[2-(2-methylphenyl)benzoyl]piperidin-4-yl}methanol
1-[7-(1-benzothiophen-3-yl)-9-(pyridin-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
1-{9-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]-3-azaspiro[5.5]undecan-3-yl}ethan-1-one
5-(naphthalen-2-yl)-3-[4-(pyridin-2-yl)piperazin-1-yl]-1,2,4-triazine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-methyl-4-phenylpyrimidine-5-carboxamide
7-(3,6-dimethylpyrazin-2-yl)-4-(3-fluoropyridine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S,4S)-N-ethyl-4-[3-(4-fluorophenyl)benzamido]-1-methylpyrrolidine-2-carboxamide
3-tert-butyl-1-methyl-4-(1-phenyl-1H-pyrazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[1-(2-fluorophenyl)-5-[(2S)-1-methanesulfonylpyrrolidin-2-yl]-1H-1,2,4-triazol-3-yl]acetamide
4-[(3,4-difluorophenyl)methyl]-N-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]piperazine-1-carboxamide
N-{[3-(dimethylamino)thiolan-3-yl]methyl}-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-N-(pyridin-3-ylmethyl)piperazine-2-carboxamide
(1-{[(4-methoxy-4-methylpentan-2-yl)amino]methyl}cyclopentyl)methanol
7-cyclohexyl-2-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-[1-(1H-indazole-3-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
1-methyl-4-(1,3-thiazol-4-ylmethyl)-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
3-{[1-(2-chlorobenzoyl)pyrrolidin-3-yl]methyl}benzoic acid
N-{[7-(2,6-dimethylhept-5-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine-4-carboxamide
2-methanesulfonamido-N-[(3R,4S)-1-(2-methoxyethyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
7-methanesulfonyl-4-methyl-2-[4-(2-methylpiperidine-1-carbonyl)piperidin-1-yl]quinazoline
(1R,5R)-N,N-dimethyl-6-[(5-methylfuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-(1,4-oxazepane-4-sulfonyl)-N-pentylbenzamide
methyl 4-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-4-oxobutanoate
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2,3-dihydro-1H-indene-1-carboxamide
2-{1-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}pyridine
[4-({1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-{2-[({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]ethyl}methanesulfonamide
methyl 2-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanoate
1-(3-fluoropropyl)-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-oxoethyl}-5-methyl-2,3-dihydro-1H-indol-2-one
N2,N2-dimethyl-N4-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
(1S,5R)-3-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
9-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-6-oxa-9-azaspiro[4.5]decane
4-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
N-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-difluorobenzamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}acetamide
2-(2-aminoethyl)-N-[2-(dimethylamino)ethyl]-5,6-dimethyl-N-(oxolan-2-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
N-[3-(3-fluorophenyl)phenyl]-1-[(trimethylpyrazin-2-yl)methyl]piperidine-4-carboxamide
methyl 3-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]benzoate
4-(1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carbonyl)morpholine
3-[2-({[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-1,3-oxazolidin-2-one
1-cyclopentyl-4-[3-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidine
2-(3-fluorophenyl)-N-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-6-ethyl-N,2-dimethylquinoline-4-carboxamide