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1-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
2-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-5-methoxy-4H-pyran-4-one
4-(1-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1H-1,2,3-triazol-4-yl)quinoline
4-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}-2,1,3-benzoxadiazole
3-[(2R,3R,6R)-5-(5-propyl-1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[(5-methoxy-1H-indol-2-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-{1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]-4-(2-phenylethyl)piperazin-2-one
5-{[4-(benzenesulfonyl)piperazin-1-yl]methyl}-2,1,3-benzothiadiazole
1-(4-fluoro-2-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}phenyl)-1H-pyrazole
3-(1H-imidazol-2-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzamide
3-[2-({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-1,3-oxazolidin-2-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(oxolan-3-ylmethyl)benzamide
1-{1-[6-(1-benzofuran-2-yl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
1-methyl-N-{3-[5-methyl-4-({[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}piperidine-3-carboxamide
methyl 5-[2-(thiophene-2-sulfonamido)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-(4-{[2-(3,4-difluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenoxy)ethan-1-ol
2-methyl-5-(propan-2-yl)-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(3-methylpyrazin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-[methyl(2-phenylethyl)amino]-N-[1-(pyrimidin-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}pyrazolo[1,5-a]pyridine-7-carboxamide
1-(naphthalen-1-ylmethyl)-N-[1-(pyridin-4-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
{1-[(2,5-dimethyl-1H-indol-3-yl)methyl]-3-[(3-methoxyphenyl)methyl]piperidin-3-yl}methanol
2-ethyl-N-(furan-2-ylmethyl)-7-(2-methoxybenzamido)-N,1-dimethyl-1H-1,3-benzodiazole-5-carboxamide
4-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-ethyl-5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
N-[2-(3-methoxyphenyl)-1-{1-[3-(4-methylphenyl)propanoyl]piperidin-4-yl}ethyl]-N,3-dimethylbutanamide
1-[4-(2-methoxypyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-2,2-diphenylethan-1-ol
N-[(2,3-dimethoxyphenyl)methyl]-6-methoxypyrimidin-4-amine
1-(2-{[(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
[4-(2-phenoxyethyl)-1-(quinolin-2-yl)piperidin-4-yl]methanol
N-benzyl-N-butyl-1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1-(pyridin-2-yl)piperidine-3-carboxamide
methyl 3-[(2-chlorophenyl)methyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(1-carbamoylcyclopentyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-(cyclohexylmethyl)-5-{[(1-hydroxycyclohexyl)methyl]amino}-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-{1-[4-(ethylamino)pyrimidin-2-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
ethyl 3-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxylate
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1,3-dimethyl-1H-indole-2-carboxamide
2-[5-(3-methoxyphenyl)-1H-indol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
1-cyclohexyl-4-(2,6-difluoro-3-methoxybenzoyl)-1,4-diazepane
2-(piperidin-1-yl)-5-{[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidine
5-[1-(6-fluoro-4-methylquinazolin-2-yl)piperidine-4-carbonyl]-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
[(5-ethylpyridin-2-yl)methyl](pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
1-{4-[(butylamino)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N'-(2,4-dimethylphenyl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]propanediamide