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1-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]-2-methoxyethan-1-one
2-(1-benzyl-4-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
N-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)acetamide
1-(6-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-3-(1,2,3-thiadiazol-5-yl)urea
N5-[2-(1,3-thiazol-4-yl)ethyl]-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-(1,2-oxazol-3-ylmethyl)-5,5-diphenylpiperidin-2-one
6-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1,3-benzothiazole
[(3R,4R)-1-(6,8-difluoro-2-methylquinolin-4-yl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3-methyl-1-{2-[2-(pyridin-2-yl)ethyl]phenyl}urea
2-(5-fluoro-2-methylphenyl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
3-({4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)phenol
5-{[2-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-1H-imidazol-1-yl]methyl}-N,N-dimethylfuran-2-carboxamide
{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-methoxybutanamide
N-methyl-N-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)thian-4-amine
methyl 1-({4-[3-(2-chlorophenyl)propanoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
(3R,4S)-1-(5,6-dimethylpyrazin-2-yl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
2,6-dimethyl-5-{2-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
1-(6-hydroxy-4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)propanamide
2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-3-carboxamide
4-[4-(3-chlorophenoxy)piperidine-1-carbonyl]-1-ethylpyrrolidin-2-one
3-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
5-(dimethylamino)-2-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-2,3-dihydropyridazin-3-one
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-3-(methylsulfanyl)-N-(oxolan-2-ylmethyl)propanamide
1-[(4aR,8aS)-1-(furan-2-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-(4-methoxyphenyl)ethan-1-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide
4-(2,5-dimethylphenyl)-7-(2-oxopyrrolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
8-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
9-(2-hydroxyethyl)-1-methyl-4-(1H-1,2,3-triazole-5-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(4-{1-[methyl(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-2-(phenylsulfanyl)ethan-1-one
1-(furan-2-ylmethyl)-1-[2-(morpholin-4-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)urea
1-(1-benzothiophen-2-ylmethyl)-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
methyl 3-[(3-hydroxypropyl)[(5-methylthiophen-2-yl)methyl]carbamoyl]benzoate
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)propanamide
4-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
2-{[(5-methylpyrazin-2-yl)methyl]amino}-N-[1-(4-propylphenyl)ethyl]acetamide
3-methyl-N-[(3S)-2-oxoazepan-3-yl]-N-({4-[3-(pyridin-3-yl)propoxy]phenyl}methyl)thiophene-2-carboxamide
N-methyl-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]acetamide
3-({[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}amino)-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
6-ethoxy-2-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}quinoline
2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
1-(2-aminoethyl)-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
6-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
5-butyl-1'-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-ethyl-5-oxo-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]pyrrolidine-3-carboxamide
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}pyridine
1-[(4-fluorophenyl)methyl]-4-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}piperazin-2-one
7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-4-[(3,4,5-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine