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2-[(3-chlorophenyl)methyl]-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1,3-benzoxazole-6-carboxamide
1-(2-propyl-1,3-thiazole-4-carbonyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-methyl-5-phenyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
3-(4-chloro-2-methylbenzoyl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
(2R,6R)-1-[(4-methanesulfonylphenyl)methyl]-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
3-[2-amino-4-methyl-6-({2-[(3-methylpyridin-4-yl)amino]ethyl}amino)pyrimidin-5-yl]propanoic acid
2-(4-methoxyphenyl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-methyl-N-[(3R)-piperidin-3-yl]-1H-1,3-benzodiazole-5-carboxamide
2-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-5-methoxy-4H-pyran-4-one
5-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-3,4-dihydropyrimidin-4-one
1-(1-{6-[6-(dimethylamino)pyridin-3-yl]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
6-tert-butyl-N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(1,2-dihydroxyethyl)-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-phenoxyethan-1-one
2-{1-benzyl-4-[(3-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-{[1-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)pyrrolidin-3-yl]methyl}benzoic acid
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[(3-methoxyphenyl)methyl]benzamide
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)benzamide
1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2,2-diphenylethan-1-one
2-{1-butyl-5-[6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidin-5-yl]-1H-1,2,4-triazol-3-yl}acetamide
1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
1-ethyl-N-[3-(methylsulfanyl)propyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
2-[4-(1-{4-[3-(hydroxymethyl)piperidine-1-carbonyl]phenyl}piperidin-4-yl)piperazin-1-yl]phenol
2-(6-chloro-3-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}imidazo[1,2-a]pyridine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline
9-({3-ethoxy-4-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-1,4,9-triazaspiro[5.5]undecan-5-one
5,6,7-trimethoxy-4-(1-phenyl-1H-pyrazol-5-yl)-1,2,3,4-tetrahydroquinolin-2-one
1-methyl-N-{[8-(3-phenylbutyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-pyrazole-3-carboxamide
(3aS,6aR)-N-cyclohexyl-3-[(3,4-dimethoxyphenyl)methyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
N-ethyl-2-methyl-N-[2-(4-methylpiperazin-1-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
3-{3-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]propyl}-3,4-dihydroquinazolin-4-one
2-{1-[(3-fluorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-(2-methoxyethyl)-1H-imidazole
4-(2-methylpropyl)-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{2-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
5-methyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-2,3-dihydro-1H-indole-2-carboxamide
6-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]pyridine-3-carboxylic acid
1-(1-propanoylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
(1S,5R)-3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
4-{[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]amino}-2-methoxypyridine-3-carbonitrile
N-(1-{7-[(3-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
N-(2-methylpropyl)-1-[1-(pent-4-enoyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
3-ethoxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
(5S,9aS,9bS)-5-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-{3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidine-1-carbonyl}pyrazine
5-(2-{2-[(2,6-diaminopyrimidin-4-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-pyrazol-1-yl)propan-1-one
4-[(2R)-2-[(2-amino-5-methylpyrimidin-4-yl)amino]-3-hydroxypropyl]phenol
1-[(2S)-2-(7-{[4-(benzyloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)pyrrolidin-1-yl]ethan-1-one