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1-{4-[(4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperazin-1-yl}ethan-1-one
N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-3-(4-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
(1R,5S,6R)-3-[(8-chloroquinolin-2-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
methyl (2S,4S)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-{2-[4-(trifluoromethyl)phenyl]benzamido}pyrrolidine-2-carboxylate
2-chloro-N-[1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
1-(4-{[2-(2-chloro-6-methylphenoxy)ethyl]amino}piperidin-1-yl)ethan-1-one
3-(2-methoxyphenyl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]propanamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
(1R,5S,8S)-8-methoxy-3-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-azabicyclo[3.2.1]octane
[(2,2-dimethyloxan-4-yl)methyl](ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
3-methoxy-N-{1-[7-(quinolin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
2-[3-(2-methyl-1H-imidazol-1-yl)propanamido]-N-[2-(morpholin-4-yl)ethyl]benzamide
2-{4-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[(3-methylpyridin-4-yl)methyl]benzamide
2-(2-hydroxyethyl)-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-methyl-1H-imidazol-2-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
3-benzyl-4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]-1-(4-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N3-cyclooctyl-N5-(furan-2-ylmethyl)-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(1-benzofuran-3-carbonyl)-4-cyclohexylpiperazine
2-[1-(1-methyl-1H-indole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
(1R,5R)-N,N-dimethyl-6-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(4aS,8aR)-6-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
N-{1-[1-(4-tert-butylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
2-methoxy-N-{1-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
5-(morpholine-4-carbonyl)-2-(phenoxymethyl)pyrimidin-4-ol
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-ethylbenzamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)cyclohex-3-ene-1-carboxamide
N-({7-[(2,3,6-trifluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzenesulfonamide
1-[2-(4-fluorophenoxy)ethyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
2-{[1-(1H-pyrazol-1-yl)propan-2-yl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[3-(4-fluorophenyl)propyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
2-({[(3R,4R)-1-(8-fluoroquinoline-2-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
4-(4-chlorophenoxy)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
1'-cyclopropanecarbonyl-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-({[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)amino)-1-phenylethan-1-ol
3-({[7-fluoro-5-(3-fluoro-4-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
N4-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-N2,6-dimethylpyrimidine-2,4-diamine
1-[2-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
1,3,6-trimethyl-5-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-fluoro-N4,N4-dimethyl-N2-[2-(thiophen-2-yl)ethyl]pyrimidine-2,4-diamine
1-benzyl-5-{[(3,4-difluorophenyl)methyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-(2-fluoro-6-methoxyphenoxymethyl)-3-(4-methoxyphenyl)-1,2,4-oxadiazole
3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[3-(propan-2-yloxy)propyl]propanamide
5-{2-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
(2S,4R)-4-amino-N-methyl-1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrrolidine-2-carboxamide
2-amino-4-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
1-(3-methoxyphenoxy)-3-[2-(pyridin-4-yl)-1H-imidazol-1-yl]propan-2-ol