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3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(4-methylphenyl)ethyl]propanamide
N-(4-fluoro-2-methylphenyl)-2-[(5-methyl-1-propyl-1H-pyrazol-4-yl)formamido]propanamide
6-methyl-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-2-(pyridin-3-yl)pyrimidin-4-amine
2-(pyrrolidin-1-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
N-[2-(2-fluorophenyl)-2-hydroxyethyl]-4-(piperidin-1-ylmethyl)benzamide
7-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
(2S)-1-[4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanoyl]pyrrolidine-2-carboxamide
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-5-(naphthalen-2-yl)-1,2,4-triazin-3-amine
6-methyl-5-{5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
(4aS,8aR)-1-(4-hydroxybutyl)-6-[4-(1H-pyrazol-4-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
3-[(5-chlorothiophen-2-yl)methyl]-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-[4-(5-propyl-1,3,4-oxadiazol-2-yl)-1,4-diazepan-1-yl]ethan-1-one
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{1-benzyl-4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-2-(pyrrolidin-1-yl)benzamide
4-(5-methylpyridin-2-yl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-ol
1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-2-(3,4,5-trimethoxyphenyl)ethan-1-one
N4-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-5,6-dimethylpyrimidine-2,4-diamine
1-(3-{4-[({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)amino]piperidin-1-yl}phenyl)imidazolidin-2-one
N-(1-benzothiophen-2-ylmethyl)-2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
(2R,3R)-1'-(5-chloropyridin-2-yl)-3-(2,5-dihydro-1H-pyrrol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
8-[(6-methylpyridin-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
5-[(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-2-methoxyphenol
methyl 1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxylate
8-(5-acetylpyridin-2-yl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-N-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
2-[5-(oxan-3-ylmethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]benzoic acid
N-[cyclopropyl(4-methoxyphenyl)methyl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
(4aS,7aR)-1-[5-(methoxymethyl)furan-2-carbonyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-chlorophenyl)-4-(2-hydroxy-4-methylbenzoyl)-5-methylpiperazin-2-one
2-(4-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
1-{3-[2-(3-fluorophenyl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
2-(3-cyclopentyl-5-{[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl)acetic acid
3-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-1-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)urea
2-oxo-6-phenyl-N-[2-(1,3-thiazol-4-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
3-(2,5-dimethylbenzoyl)-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-[(1-cyclohexylpiperidin-4-yl)oxy]-N-(pyridin-2-ylmethyl)benzamide
1-(4-{[3-(cyclopentylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}thiophen-2-yl)ethan-1-one
N-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-2-(pyridin-2-yl)pyrrolidine-1-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N,3,6-trimethyl-1-benzofuran-2-carboxamide
2-[(2-fluorophenyl)methyl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-benzoxazole-6-carboxamide
2-{4-[4-(3,3-difluoropiperidine-1-carbonyl)-6-ethylquinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
1-(2,2-dimethylpropyl)-3-hydroxy-3-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)piperidin-2-one
2,3-dimethyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-indole-7-carboxamide
N-[(1R,2R)-2-(dimethylamino)-2,3-dihydro-1H-inden-1-yl]-4-(3-hydroxy-3-methylbutyl)benzamide
N-butyl-N-methyl-2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)acetamide