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4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-5-methyl-3-phenyl-1,2-oxazole
N-[1-(2,5-difluorophenyl)cyclopropyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)morpholine-2-carboxamide
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-methyl-4-{3-[(1-methylpiperidin-4-yl)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}pyridin-2-amine
4-{1-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-dihydrophthalazin-1-one
(3S,4R)-4-(hydroxymethyl)-1-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)piperidin-3-ol
N-benzyl-N-ethyl-4-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]pyridine-2-carboxamide
N-{[(2S,4S)-4-fluoro-1-(propane-2-sulfonyl)pyrrolidin-2-yl]methyl}pentanamide
{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
2-(1-methyl-4-{1-[3-(2-methylphenyl)phenyl]piperidin-4-yl}piperazin-2-yl)ethan-1-ol
3-{[(2-chlorophenyl)formamido]methyl}-N-(2-methoxyphenyl)piperidine-1-carboxamide
5-methyl-5-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
7-fluoro-N-(2-methoxyethyl)-2-methyl-N-propylquinoline-4-carboxamide
(2E)-3-(4-methoxyphenyl)-1-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)prop-2-en-1-one
N-[3-(4-{[2-(2,6-difluorophenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-3-(pyridin-3-yl)propanamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylpent-4-enamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide
2-methyl-5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-3,4-dihydropyrimidin-4-one
6-[4-(2-methoxyethyl)piperazin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
N-{4-[(2S)-2-amino-3-(1H-imidazol-4-yl)propanamido]-2-methoxyphenyl}butanamide
3-(2-fluorophenyl)-N-methyl-3-phenyl-N-(pyridin-3-ylmethyl)propanamide
1-[(2E)-3-phenylprop-2-en-1-yl]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(2S,4S)-4-amino-N-ethyl-1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)pyrrolidine-2-carboxamide
1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N-cyclopropyl-5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
1-[2-(2-phenylphenyl)-1H-imidazol-1-yl]propan-2-ol
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-2-(propan-2-yloxy)propanamide
N-methyl-4-(1-phenyl-1H-pyrazol-4-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrimidin-2-amine
1-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
5-fluoro-1-methyl-2-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}-1H-indole
1-(2,5-dimethylphenyl)-4-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
2-amino-4-cyclopropyl-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
{2-methoxy-5-[1-(3-methylbutyl)-1H-pyrazol-4-yl]phenyl}methanol
3-chloro-N-[2-(dimethylamino)ethyl]-4-[(1-{spiro[2.3]hexane-1-carbonyl}piperidin-4-yl)oxy]benzamide
2-cyclohexyl-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1,3-benzoxazole-6-carboxamide
1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
7-(2-cyclohexylethyl)-2-cyclopentanecarbonyl-2,7-diazaspiro[4.5]decan-6-one
N-[(3-methylpyridin-2-yl)methyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
2-amino-4-{3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-7-methyl-5H,7H-furo[3,4-b]pyridine-3-carbonitrile
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine
2-[4-(2-fluorophenyl)piperazin-1-yl]-N-(1-hydroxypropan-2-yl)-6-(2-methoxyphenyl)pyridine-3-carboxamide
4-fluoro-N-{3-[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]-3-oxopropyl}benzamide
3-{1-[(5-ethylfuran-2-yl)methyl]piperidin-2-yl}propan-1-ol
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
1-[4-(2-butyl-1,3-benzoxazole-5-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-[(3S)-2-oxoazepan-3-yl]-1,2-oxazole-3-carboxamide
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-(2-methyl-4-phenylpiperazin-1-yl)propan-1-one