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5-cyclobutanecarbonyl-1'-[(6-methylpyridin-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(3,4-dimethylphenyl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-2-(1H-pyrazol-1-yl)acetamide
4-{2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyridine
N-cyclopropyl-3-{[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]sulfamoyl}benzamide
N-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl}-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
3-[methyl(propan-2-yl)amino]-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}propanamide
(1-{1-[(1-benzyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanamine
N-(2-methylquinolin-8-yl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
3-methoxy-N-{2-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1,2,3,4-tetrahydroisoquinolin-7-yl}propanamide
2-methoxy-1-[1'-(1H-pyrrole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
5-methyl-N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-(4-methoxyphenyl)-4-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}piperazine
3-[3-(1H-pyrazol-3-yl)phenyl]thiophene-2-carbonitrile
3-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
N2,N2-dimethyl-N4-[1-(4-methylpyridin-2-yl)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
2,6-dihydroxy-N-[1-(pyridin-3-yl)pentyl]benzamide
5-{4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-N-methylpyrimidin-2-amine
1-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
[(3R,4R)-1-(1-benzofuran-5-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
5-benzyl-4-(2-ethoxyacetyl)-1-(4-methylphenyl)piperazin-2-one
2-{1-[(2-ethoxyphenyl)methyl]-4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]acetamide
{1-methyl-5-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
2-benzyl-8-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-2,8-diazaspiro[5.5]undecane
{3-[(4-fluorophenyl)methyl]-1-[(4-methoxyphenyl)methyl]piperidin-3-yl}methanol
1-(4-methyl-1,3-oxazole-5-carbonyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
2-tert-butyl-4-hydroxy-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]pyrimidine-5-carboxamide
8-(5-ethyl-1,3-oxazole-4-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-1-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidine-2-carboxamide
4,6-dimethyl-2-oxo-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
[4-(2-phenoxyethyl)-1-(quinoline-8-sulfonyl)piperidin-4-yl]methanol
1-[(2-methylpyrimidin-5-yl)methyl]-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide
1-{1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
6-{1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-4-yl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
2-(2,2-dimethylpropanamido)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,5-dimethylthiophene-3-carboxamide
3-(3,4-dimethoxyphenyl)-1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]propan-1-one
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
2-{[(3R,5S)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidin-3-yl]sulfanyl}-1H-1,3-benzodiazole
2-{[(1-ethylpiperidin-4-yl)methyl](methyl)amino}-1-phenylethan-1-ol
(2R)-1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-2-phenylethan-1-one
6-amino-1-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}hexan-1-one
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[4-(2-phenoxyethyl)piperazin-1-yl]ethan-1-one
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
1-(4-methyl-1,2,5-oxadiazol-3-yl)-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperazine
(3R,4R)-1-(1-benzofuran-2-ylmethyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol