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7-(2-hydroxyethyl)-2-(2-methoxypyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(3S,4S)-1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-4-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyrrolidin-3-ol
2-[(2,6-difluoro-4-methoxyphenyl)methyl]-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
N-(1-cyclopropanecarbonylpiperidin-3-yl)-2-fluoro-5-sulfamoylbenzamide
1-[2-methoxy-4-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
N-(4-chloro-3-methylphenyl)-4-[hydroxy(pyridin-2-yl)methyl]piperidine-1-carboxamide
3-(2-phenylethyl)-5-(piperidin-4-yl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
(3S,4S)-1-[5-(2-chlorophenyl)furan-2-carbonyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
1-[3-methyl-4-(pyridine-3-amido)phenyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxylic acid
(2S,4R)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-[(2-methoxynaphthalen-1-yl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(2-phenylpropyl)piperidine-4-carboxamide
[(5-methoxy-3-methyl-1H-indol-2-yl)methyl](methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-3-fluoro-2-methoxybenzamide
5-[(2-chlorophenyl)methyl]-5-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
9-(6-chloropyridazin-3-yl)-3-oxa-9-azaspiro[5.5]undecane
N-cyclobutyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
1-{[4-(difluoromethoxy)phenyl]methyl}-N-[2-(dimethylamino)ethyl]-N-methylpiperidin-3-amine
N-cyclopropyl-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-(diphenylmethyl)-N-methyl-N-(oxan-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1-phenyl-1H-1,2,3-triazole-5-carboxamide
{1-[(2-chloro-6-fluorophenyl)methyl]-3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
N-[(2-fluorophenyl)methyl]-1-methyl-5-{[2-(pyridin-2-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3S,9aR)-3-[(benzyloxy)methyl]-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(oxolan-2-ylmethyl)-2-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[(3R,5S)-5-[(2,1,3-benzoxadiazol-5-ylmethyl)carbamoyl]pyrrolidin-3-yl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
2-[(2-butylpyrrolidin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylthiophene-3-carboxamide
1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3-(4H-1,2,4-triazol-3-yl)piperidine
2-cyclopentyl-N-cyclopropyl-N-({3-[(2-fluorophenyl)methoxy]phenyl}methyl)acetamide
2-({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)propan-1-ol
(1S,5R)-6-(1,3-thiazol-4-ylmethyl)-3-{2-[(trifluoromethyl)sulfanyl]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-2-methoxyphenol
N-(2,3-dihydro-1H-inden-2-yl)-2-(furan-2-yl)-2-oxoacetamide
1-[1-(3-methylbenzoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(thiophen-2-ylmethyl)pyrimidin-2-amine
5-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-3-[3-(dimethylamino)propyl]-5-[(2-methylphenyl)methyl]imidazolidine-2,4-dione
2-[(4aR,7aS)-4-[2-(6-methylpyridin-2-yl)ethyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
(2S)-2-({[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)-4-methylpentanamide
2-(pyridin-2-ylmethyl)-8-[2-(pyrrolidin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[(2-chlorophenyl)methyl]-N-cyclopropyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
methyl 4-[4-(1H-pyrazol-1-yl)phenyl]-1H-pyrrole-2-carboxylate
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-methoxyethan-1-one
methyl (2S)-1-[3-(3,4-dimethylbenzoyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]pyrrolidine-2-carboxylate
1-{7-methylthieno[3,2-d]pyrimidin-4-yl}-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
6-(methoxymethyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidin-4-amine
5-({[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]amino}methyl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(4-methyl-1H-imidazol-5-yl)methyl]amine
N-({8-[(2,4-dimethylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
3-[4-(dimethylamino)phenyl]-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide