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1-[(4aR,8aR)-4a-hydroxy-7-methanesulfonyl-decahydro-2,7-naphthyridin-2-yl]-2-(2-fluorophenyl)ethan-1-one
1-ethyl-N-[(1-ethylpiperidin-3-yl)methyl]-5-(2-methoxyacetamido)-N-methyl-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carboxamide
1-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
3-{2-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3-hydroxypyrrolidin-3-yl)methyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
N,N-dimethyl-6-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyrazin-2-amine
N-(1-phenylethyl)-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[1-(methoxymethyl)cyclopentyl]quinoxaline-6-carboxamide
4-chloro-N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-ethyl-1,2,3-thiadiazole-5-carboxamide
N-({3-methyl-7-[4-(methylsulfanyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)methanesulfonamide
N-({1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}methyl)-2-(2-methoxyphenoxy)acetamide
1-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-3-ol
(1R,3S)-3-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-N,N,2,2,3-pentamethylcyclopentane-1-carboxamide
methyl 3-{[3-(2-hydroxyethoxy)phenyl]methyl}-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-N-(3-chloro-4-fluorophenyl)propanamide
5-{1-[1-(pyridin-4-yl)propyl]-1H-imidazol-2-yl}-2,1,3-benzothiadiazole
{3-[(dimethyl-1,2-oxazol-4-yl)methyl]-9-[(1-methyl-1H-imidazol-5-yl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
3-(3-hydroxyquinoxalin-2-yl)-N-methyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}propanamide
4-[1-(9H-fluoren-2-ylmethyl)azetidin-3-yl]pyridine
1-(furan-2-ylmethyl)-4-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperazine
1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-2-(1-methyl-1H-imidazol-2-yl)piperidine
6-[4-(1-cyano-1-methylethyl)phenyl]pyrazine-2-carboxylic acid
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-[(6-methylpyridin-2-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
1-(2-{[(5-phenyl-1,2,4-oxadiazol-3-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
(3R)-1-[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidin-3-ol
2-{4-[(2-chlorophenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-methyl-N-[(5-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}furan-2-yl)methyl]methanesulfonamide
2-amino-6-[1-(3-chlorophenyl)-1H-pyrazol-4-yl]-4-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
5-methyl-1'-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-cyclopentyl-6-oxo-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
N-[(3-methoxyphenyl)methyl]-N-methyl-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decane-8-carbonyl}benzonitrile
N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-3-{[4-(propan-2-yloxy)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-[(2-chlorophenyl)methyl]-N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3R,4R)-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
4-(1-{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-5-methylpyrimidine
1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-3-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
6-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-N-(propan-2-yl)pyrimidin-4-amine
1-[4-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
(1R,7S)-3-(pyridin-3-ylmethyl)-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-3-(4-chloro-1H-pyrazol-1-yl)propan-1-one
4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
(1S,9aR)-1-[(4-phenylpiperidin-1-yl)methyl]-octahydro-1H-quinolizine
N-(1,3-benzoxazol-2-ylmethyl)-4-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
(2S,4S)-4-amino-N,N-diethyl-1-(5-hydroxypyrazine-2-carbonyl)pyrrolidine-2-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one