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{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[2-(4-phenylpyrimidin-2-yl)ethyl]amine
N-methyl-6-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
2-{[2-(4-methoxyphenyl)piperidin-1-yl]methyl}pyridine-3-carboxylic acid
1-cyclopropyl-N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
2-(1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)-5-fluoro-1H-1,3-benzodiazole
2-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-3-methylquinoxaline
4-({2-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-ethyl-5-[4-(2-methoxyphenyl)piperazin-1-yl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-{4-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]morpholin-3-yl}acetic acid
3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-[2-(1H-pyrazol-1-yl)phenyl]urea
1-[(2-methoxyphenyl)methyl]-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
8-methoxy-5-[3-(pyrrolidin-1-yl)pyrazin-2-yl]quinoline
1-(2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carbonyl)-2-methylpiperidine-2-carboxylic acid
1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-3-phenyl-1H-pyrazole-5-carboxamide
N-(2-methoxyethyl)-4-methyl-3-{[(1,2-oxazol-3-ylmethyl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
3-(5-{[(3-hydroxypropyl)[(5-methylthiophen-2-yl)methyl]amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
1-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 6-{2-benzyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pyrimidine-4-carboxylate
5-ethyl-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N,2,3-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
2-(4-methyl-1H-imidazole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
2-[8-(2,3-dihydro-1H-inden-2-yl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
(3R,4S)-4-cyclopropyl-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-amine
2-hydroxy-4-methoxy-N-{[1-(1-methylpiperidin-4-yl)pyrrolidin-3-yl]methyl}benzamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(2-phenylethyl)piperidine
5-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-1-[(2-methoxyphenyl)methyl]-N-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
4-({5-[1-(cyclohexylmethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
4-(1,3,6-trimethyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)benzoic acid
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(quinolin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1-{1-[2-(dimethylamino)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-fluorobenzamide
2,6-dimethyl-N-[1-(thian-4-yl)piperidin-4-yl]imidazo[1,2-a]pyridine-3-carboxamide
3-(furan-2-yl)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]propanamide
2-{4-[4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]piperazin-1-yl}-1,3-benzoxazole
N-[(3-chlorophenyl)methyl]-3-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}propanamide
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-methoxypyrimidin-2-amine
2-methyl-N-[5-(morpholin-4-yl)pentyl]thieno[2,3-d]pyrimidin-4-amine
1-methyl-9-(4-methylnaphthalene-1-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
N-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-1-(oxan-4-yl)piperidine-4-carboxamide
4-[(4-fluorophenyl)methyl]-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
N-methyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
4-{5-[({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]thiophen-2-yl}-2-methylbut-3-yn-2-ol
3-({[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)propan-1-ol
2-acetamido-N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}acetamide
1-ethyl-2-(5-methyl-1-benzofuran-2-carbonyl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine
N-[4-(2-hydroxyethyl)phenyl]-4-[(3-methylpiperidin-1-yl)methyl]benzamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(pyridin-4-ylmethyl)piperidin-3-yl]propanamide