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N-{[1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
4-[4-benzyl-3-oxo-6-(pyridin-2-ylmethoxy)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
N-methyl-N-{[5-({[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amino}methyl)furan-2-yl]methyl}methanesulfonamide
4-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenol
4-(2,4-dioxoimidazolidin-1-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]benzamide
1-acetyl-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-[2-(tert-butylsulfamoyl)phenyl]pyrazine-2-carboxylic acid
(benzylsulfamoyl)(methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
N-(3,5-dimethoxyphenyl)-3-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]propanamide
4-hydroxy-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
2-[(2-fluorophenyl)methyl]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-6-carboxamide
N-{2-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]ethyl}acetamide
3-(1H-imidazol-1-ylmethyl)-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidine
N-({1-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
N-benzyl-1-methyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
[5-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)-2-ethoxyphenyl]methanol
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-5-methyl-1,3,4-oxadiazole-2-carboxamide
N-benzyl-2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]acetamide
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
(3aS,6aS)-2-methyl-5-phenylmethanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2,2-dimethyloxan-4-yl)-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
5-(morpholin-4-yl)-2-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]-2,3-dihydropyridazin-3-one
(3S,5S)-5-(cyclopropylcarbamoyl)-1-[3-(1H-indol-3-yl)propanoyl]piperidine-3-carboxylic acid
N,N-diethyl-2-{4-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}acetamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methylacetamide
N-(5-methyl-1,3,4-thiadiazol-2-yl)-4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
2-(3,4-dichlorophenyl)-4-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}morpholine
4-[(2-ethyl-1H-imidazol-1-yl)methyl]-5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazole
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-8-fluoro-4-oxo-1,4-dihydroquinoline-2-carboxamide
N-ethyl-N-methyl-6-[3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxamide
N-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(2-methoxypyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]methyl}-1H-indole
[(3R,4R)-1-[3-(dimethylamino)benzoyl]-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
N-{3-[1-(3-chlorophenyl)-1H-1,2,4-triazol-5-yl]propyl}acetamide
2-(1-{1-oxaspiro[4.4]nonan-3-yl}-1H-imidazol-2-yl)pyridine
2-(2-fluorophenyl)-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]acetamide
1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(dimethyl-1,2-oxazol-4-yl)-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
N-{2-methyl-1-[3-(morpholin-4-yl)piperidin-1-yl]-1-oxopropan-2-yl}thiophene-2-carboxamide
1-[2-(2-ethylphenyl)pyridine-4-carbonyl]-4-methylpiperazine
5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(2-methoxy-5-methylphenyl)-2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]acetamide
5-(2,4-dimethoxyphenyl)-N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-1,2,4-triazin-3-amine
2-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
1-(4-{[(3-fluoro-4-methylphenyl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
5-{1-[(6-chloro-4-oxo-4H-chromen-3-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
(1-methyl-1H-imidazol-2-yl)({1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-4-yl})methanol
5-{2-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione