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{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-[(3-methoxyphenyl)methyl]piperidin-3-yl}methanol
ethyl 4-(2-phenoxyethyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-4-carboxylate
N-{[3-(difluoromethoxy)phenyl]methyl}-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
N-methyl-3-(1-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperidin-3-yl)-N-(1-methylpiperidin-4-yl)propanamide
1-[(2-methyl-1H-imidazol-4-yl)methyl]-4-(1H-pyrazol-1-ylmethyl)piperidine
(1S,5R)-6-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(3,4-dimethoxyphenyl)-1-(9H-purin-6-yl)piperidin-3-amine
N-(2-methyl-1-{7-[(6-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)methanesulfonamide
N-[(3-methoxyphenyl)methyl]-N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
7-(4-tert-butylbenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(1R,5S,6R)-3-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-N-(pyridin-2-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
2-(3-methyl-1H-pyrazol-1-yl)-1-{3-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one
ethyl 3-[(2-fluorophenyl)methyl]-1-[4-(1H-imidazol-1-yl)benzoyl]piperidine-3-carboxylate
ethyl 1-methyl-5-{1-[3-(trifluoromethyl)phenyl]propan-2-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[1-(cyclohexylmethyl)-4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperazin-2-yl]ethan-1-ol
methyl 3-(6-methylpyridine-3-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(4-fluorobenzoyl)-5-methyl-1-(3-methylphenyl)piperazin-2-one
1-[(2S)-pyrrolidine-2-carbonyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-[(1-acetylpiperidin-4-yl)oxy]-N-(2-hydroxyethyl)-5-methoxy-N-(thiophen-2-ylmethyl)benzamide
9-(2,3-dimethyl-1H-indole-7-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-(piperazin-1-yl)ethan-1-one
N-(2-{[2-(4-fluorophenoxymethyl)-4-hydroxypyrimidin-5-yl]formamido}ethyl)acetamide
(dicyclopropylmethyl)({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)methylamine
N-cyclopentyl-2-(2-methyl-1,3-thiazol-4-yl)-N-(3-phenylprop-2-yn-1-yl)acetamide
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amine
(4aS,8aR)-6-[(2-methyl-1H-imidazol-4-yl)methyl]-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
{[6-methyl-2-(prop-2-en-1-yloxy)quinolin-3-yl]methyl}(oxolan-2-ylmethyl)amine
2-[(2S)-2-aminobutanoyl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-ethyl-6-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxamide
1-(2-methoxyphenyl)-4-[2-(oxolan-3-yl)ethyl]piperazin-2-one
3-(3-methoxyphenyl)-N-[3-(oxolan-3-yl)propyl]-1H-pyrazole-5-carboxamide
8-[2-(adamantan-1-ylsulfanyl)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-1-ethyl-3-methylpiperidine-3-carboxamide
2-amino-6-ethyl-4-[2-(morpholin-4-yl)pyrimidin-5-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-[7-(1,3-benzothiazol-2-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]acetamide
[5-(1-{[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]pyridin-2-amine
2-{[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]methyl}-3-(furan-2-yl)propan-1-ol
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
N3-ethyl-1-(2-methoxyethyl)-N3-(2-methylprop-2-en-1-yl)-4-oxo-N5-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-[(3S,4R)-1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-(2-aminoethyl)-N-[2-(2-chloro-6-fluorophenyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-phenylbutanamide
1-benzyl-3-(2-methylpropyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-3-(1-methylpiperidin-4-yl)propan-1-one
2-({[2-(4-fluorophenyl)ethyl]amino}methyl)-4-(pyrazin-2-yl)phenol
{4-[(3-methoxyphenyl)methyl]-1-(2-methyloxane-2-carbonyl)piperidin-4-yl}methanol