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{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylpyridin-2-yl)methyl]amine
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
8-(2-amino-9H-purin-6-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[3-(ethylsulfanyl)propanoyl]pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
4-{5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}thiomorpholine
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-(cyclohex-1-en-1-yl)ethan-1-one
[(1-{[1-(6-chloropyridin-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]urea
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]oxane-4-carboxamide
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-2-(1-ethylpiperidin-4-yl)acetamide
(4aR,7aS)-1-ethyl-4-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,6-dimethyl-5-{2-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)acetamide
N-(2-{7-[3-(5-methylfuran-2-yl)butyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
(1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-3-(2-methoxyethyl)piperidin-3-yl)methanol
(1S,6R)-9-{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3-methyl-3,9-diazabicyclo[4.2.1]nonane
1-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5,5-diphenylpiperidin-2-one
N-(dicyclopropylmethyl)-2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-methylacetamide
(1R,5R)-6-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-({1-[(2S)-2-aminopentanoyl]piperidin-4-yl}methyl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]amine
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-[(3-methylphenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
3-(1-benzothiophen-2-ylmethyl)-9-methoxy-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
(2S)-4-methyl-2-phenyl-1-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}piperazine
3-(1-cyclohexyl-1H-pyrazol-5-yl)-1-(2-methoxyethyl)-1-(pyridin-3-ylmethyl)urea
(1S,5R)-6-(4-methoxy-3,5-dimethylbenzenesulfonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-(5-methyl-1H-pyrazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(3-methoxybenzoyl)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
N-[(3S,4R)-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2-{[(3S,5S)-5-[4-(adamantan-2-yl)piperazine-1-carbonyl]-1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidin-3-yl]sulfanyl}-4-methylpyrimidine
1-[3-(1H-imidazol-2-yl)propyl]-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
2-(5-fluoro-2-methylphenyl)-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-[2-(thiomorpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
2-[4-(1-ethyl-1H-1,2,4-triazol-5-yl)-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl]acetic acid
1-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}ethan-1-one
2-chloro-4-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]phenol
2-(2-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]methyl}-6-methoxyphenoxy)propanoic acid
2-{1-cyclohexyl-5-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]-1H-1,2,4-triazol-3-yl}acetamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2,3-dimethoxyphenyl)methyl]acetamide
2-butyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,3-benzoxazole-5-carboxamide
6,7-dimethoxy-2-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1,2,3,4-tetrahydroisoquinoline
N-ethyl-2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
2-(3-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}phenyl)-1H-imidazole
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
(3S,4R)-1-[(4-cyanophenyl)methyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
2-[1-(2,2-dimethylpropyl)-4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[2-(4-methylphenoxy)acetyl]piperidin-4-yl}propanamide
1-{3-[(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)methyl]phenyl}ethan-1-one