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N-[(4-methoxyphenyl)methyl]-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
N-{5-[2-(3-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}-2-(oxan-4-yl)acetamide
(2S)-2-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]-2-phenylethan-1-ol
2-[4-(1-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]-N,N-dimethylacetamide
2-amino-N-cyclopentyl-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(4-methylphenyl)methyl]acetamide
5-methoxy-N-methyl-4-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-4H-pyran-2-carboxamide
1-phenyl-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(3,5-dimethylbenzoyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{2-[methyl(phenyl)amino]ethyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[5-(3-acetylphenoxymethyl)-1H-pyrazole-3-carbonyl]-2-methyl-1,4-diazepan-5-one
(2R,3S,6R)-3-phenyl-5-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-phenylpropanamide
3-[1-(1-benzyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]benzoic acid
3-(1-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1H-1,2,3-triazol-4-yl)phenol
4-[(3-methoxyphenyl)methyl]-1-{2-[3-(trifluoromethyl)phenyl]acetyl}-1,4-diazepan-5-one
N-benzyl-2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}acetamide
N-methyl-1-phenyl-N-[1-(pyrimidin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-[3-(furan-2-yl)benzoyl]-1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
4-ethyl-N-{2-[4-(propan-2-yl)morpholin-2-yl]ethyl}-1,2,3-thiadiazole-5-carboxamide
3-(3-hydroxy-2,2-dimethylpropyl)-3,4-dihydroquinazolin-4-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}acetamide
6-{10-oxo-3,9-diazaspiro[5.6]dodecan-3-yl}pyridine-3-carbonitrile
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
N-(1,3-benzothiazol-2-ylmethyl)-2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-methylacetamide
1-methyl-6-propyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(5-ethyl-1,3-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-oxo-N-[2-(propylsulfanyl)ethyl]-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
5-chloro-3-[4-(3-hydroxyphenyl)piperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
1-[(2S,6S)-6-butyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)ethan-1-one
N-(5-chloro-2-methoxyphenyl)-2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
2-(2,3-dihydro-1-benzofuran-7-yl)-2-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}acetic acid
N-[3-(morpholin-4-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl})amine
(3aS,6aS)-2-(2-methoxyethyl)-5-{[4-(trifluoromethyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-3-methyl-1-[3-(1H-pyrazol-5-yl)phenyl]urea
N-{3-methyl-4-[2-(6-methylpyridin-2-yl)-1H-imidazol-1-yl]phenyl}acetamide
methyl (2S,3S)-2-{[5-(3,4-difluorophenoxymethyl)-1,2-oxazol-3-yl]formamido}-3-methylpentanoate
5-(4-acetylphenoxymethyl)-N-cycloheptyl-1,2-oxazole-3-carboxamide
(1S,3R)-3-amino-N-[2-(benzyloxy)phenyl]cyclopentane-1-carboxamide
{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
3-methoxy-5-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}thiophene-2-carboxamide
3-[5-(1-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
1-(carbamoylmethyl)-N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-4-carboxamide
N-cyclopentyl-3-[methyl(thian-4-yl)sulfamoyl]benzamide
(1H-1,3-benzodiazol-2-ylmethyl)(butan-2-yl)(pyridin-3-ylmethyl)amine
7-fluoro-2-methyl-4-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]quinoline
2-ethyl-8-[6-(trifluoromethyl)pyridin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(2-ethylphenoxy)azetidin-1-yl]ethan-1-one