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1-methyl-4-{1-[1-(1H-pyrazole-3-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
2-hydroxy-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}acetamide
4-{4-[1-(2-methyl-1H-1,3-benzodiazol-6-yl)-1H-imidazol-2-yl]phenyl}but-3-yn-1-ol
2-(1-methyl-4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperazin-2-yl)ethan-1-ol
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-benzoxazole
3-[3-(3-chlorophenyl)pyrrolidine-1-carbonyl]-5-(2,6-difluorophenoxymethyl)-1,2-oxazole
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propan-1-one
[2-(4-methanesulfonylphenyl)-8-methylquinolin-3-yl]methanol
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(pyridin-3-ylmethyl)oxane-4-carboxamide
(2S,4R)-N,N-diethyl-1-(4-hydroxybenzoyl)-4-(2-methoxyacetamido)pyrrolidine-2-carboxamide
N-{[1-(furan-3-ylmethyl)pyrrolidin-3-yl]methyl}-1-phenylcyclopropane-1-carboxamide
3-fluoro-N-[(7-{[4-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}cyclopropanamine
4-(5-methyl-1H-pyrazole-3-carbonyl)-2-(naphthalen-1-ylmethyl)morpholine
4-[(2-methylphenyl)methyl]-1-[(3-methylthiophen-2-yl)methyl]-1,4-diazepan-5-one
2-(5-methyl-1,2-oxazol-3-yl)-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidine
3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
1-methyl-4-{[3-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-5-phenyl-1H-pyrazole
N-[2-(1H-imidazol-1-yl)propyl]-2,8-dimethylquinoline-4-carboxamide
N-ethyl-N-[(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)methyl]-2-phenoxypropanamide
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(oxolan-3-yl)benzamide
4-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-1-(3-methoxyphenyl)piperazin-2-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-phenyl-5-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-(4-methyl-2-{[3-(morpholin-4-yl)propyl]amino}pyrimidin-5-yl)ethan-1-one
N-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-1,2,3-triazole-4-carboxamide
3-[(methylsulfanyl)methyl]-1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperidine
2-[4-(oxane-2-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
N-[1-(1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2,2-dimethylpropanamide
3-methyl-5-[1-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)pyrrolidin-2-yl]-1H-1,2,4-triazole
diethyl(2-{2-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)amine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{3-[methyl(phenyl)amino]propyl}acetamide
5-[1-(1-methylpiperidine-2-carbonyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-(1-benzofuran-5-yl)-4-(dimethylamino)azepane-1-carboxamide
3-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-1-[2-(pyridin-2-yl)ethyl]urea
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2-(5-oxopyrrolidin-2-yl)acetamide
4-acetyl-N-(3-methanesulfonamido-4-methoxyphenyl)piperazine-1-carboxamide
4-({4-methyl-5-[1-(3,3,3-trifluoropropyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]pyridine-3-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N,3,6,7-tetramethyl-1-benzofuran-2-carboxamide
5-ethyl-2-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}pyridine
2-(2,3-difluorophenyl)-2-[4-(morpholin-4-yl)piperidin-1-yl]acetic acid
2-(3-hydroxypropyl)-8-(naphthalen-1-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(4aR,8aR)-2-cyclopentanecarbonyl-7-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
3-(4-methoxyphenyl)-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]propan-1-one
2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-5-methylpyrimidin-4-amine
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)propane-1-sulfonamide
1-[2-({5-propylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]imidazolidin-2-one
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2,4-dimethylpyrimidine-5-carboxamide