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5-[5-(ethoxymethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-2-(thiophene-3-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
4-[(2R,3R)-2-hydroxy-1'-(thiophene-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperazin-2-one
(3aR,5R,6S,7aS)-2-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-octahydro-1H-isoindole-5,6-diol
3-({4-[1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
6-ethyl-N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-2-methylquinoline-4-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-N-{[1-(dimethylamino)cyclohexyl]methyl}-5-methoxybenzamide
3-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-3-yl}-N-[(3,4-difluorophenyl)methyl]propanamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}furan-2-carboxamide
4-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
2-(2-fluorophenoxymethyl)-N-[(1-methylpiperidin-2-yl)methyl]-1,3-oxazole-4-carboxamide
2-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
N-(4-fluorophenyl)-1-[2-(methylsulfanyl)benzoyl]piperidin-3-amine
6-methyl-2-{1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
1-{4-[(2-methoxy-2-methylpropyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
3-{2-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)-3-(2-methoxyphenyl)pyrrolidine-2,5-dione
2-{1-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-(2-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}ethoxy)ethan-1-ol
1-[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
7-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
3,5,7-trimethyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
1-cyclopropyl-3-(2,6-dimethoxypyridin-3-yl)-1-{[4-(methylsulfanyl)phenyl]methyl}urea
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(2,3-dihydro-1H-isoindol-2-yl)-1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
[1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl](thiophen-2-yl)methanol
5-(5-methylfuran-2-yl)-3-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]-1,2,4-triazine
[2-(azepan-1-yl)ethyl](ethyl)[(1-ethyl-1H-pyrazol-4-yl)methyl]amine
N-benzyl-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
(1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-propylpiperidin-4-yl)methanol
3-(3-methoxypropyl)-1-[(3-methylpyridin-2-yl)methyl]piperidine-3-carboxylic acid
1-benzoyl-N-methyl-N-[1-(pyridin-2-yl)ethyl]piperidin-4-amine
2-({3-[3-(1,3-thiazol-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)pyridine
N-(1-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
N-(cyclopropylmethyl)-2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
N-{2-[7-(naphthalen-1-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-phenoxyacetamide
N,N-dimethyl-2-[(1S,5R)-6-[3-(thiophen-2-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
5-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
3-phenyl-5-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}-3-methylpiperazin-2-one
1-(2-methoxyphenyl)-3-{1-[1-(1-methylpiperidine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
ethyl 1-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carbonyl}piperidine-3-carboxylate
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-4-methoxy-N-(oxolan-2-ylmethyl)benzamide
N-{3-[2-benzyl-4-(2-methylphenyl)-5-oxopiperazin-1-yl]-3-oxopropyl}acetamide
N-[1-(benzenesulfonyl)piperidin-4-yl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-4-(piperidine-1-carbonyl)pyridin-2-amine
1-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}azepane
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}oxy)benzamide
N-(1-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide